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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T35567 | BIX01294 (hydrochloride hydrate) | ||
The methylation of lysine residues on histones plays a central role in determining euchromatin structure and gene expression. The histone methyltransferase (HMTase) G9a can mono- or dimethylate lysine 9 on histone 3 (H3)... | |||
T1959 | BIX-01294 trihydrochloride | BIX 01294 | Histone Methyltransferase , Autophagy |
BIX-01294 trihydrochloride is an inhibitor of G9a histone methyltransferase.In a cell-free assay, the IC50=2.7 μM for G9a histone methyltransferase. | |||
T7697 | BIX-01294 | Histone Methyltransferase , Autophagy | |
BIX-01294 is an G9a Histone Methyltransferase inhibitor(IC50 : 1.9 μM). | |||
T36779 | NG 25 (hydrochloride hydrate) | ||
NG 25 is a type II kinase inhibitor that inhibits MAP4K2 and TAK1 (IC50s = 21.7 and 149 nM, respectively).1It also inhibits the Src family kinases Src and LYN (IC50s = 113 and 12.9 nM, respectively) and Abl family kinase... | |||
T38323 | A-943931 (hydrochloride hydrate) | ||
A-943931 is a histamine H4receptor antagonist (Ki= 3.8 nM).1In vivo, A-943931 inhibits scratching induced by clobenpropit in mice (ED50= 26 μmoles/kg, i.p.). 1.Milicic, I., Witte, D.G., Miller, T.L., et al.Identification... | |||
T8404 | Kasugamycin hydrochloride hydrate | Ksg (hydrochloride hydrate) | Antibacterial , Antibiotic |
Kasugamycin hydrochloride hydrate (Ksg (hydrochloride hydrate))(Ksg) specifically inhibits translation initiation of canonical but not of leaderless messenger RNAs. Ksg inhibition is thought to occur by direct competitio... |