Powder: -20°C for 3 years | In solvent: -80°C for 1 year
XD14 is an inhibitor of BET bromodomain (Kd of 160 nM, 170 nM, 380 nM, 490 nM, 830 nM and 850 nM for BRD4(1), BRD2(1), BRD3(1), BRD3(2), BRD2(2) and BRD4(2), respectively).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 43.00 | |
5 mg | In stock | $ 98.00 | |
10 mg | In stock | $ 172.00 | |
25 mg | In stock | $ 347.00 | |
50 mg | In stock | $ 555.00 | |
100 mg | In stock | $ 783.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 116.00 |
Description | XD14 is an inhibitor of BET bromodomain (Kd of 160 nM, 170 nM, 380 nM, 490 nM, 830 nM and 850 nM for BRD4(1), BRD2(1), BRD3(1), BRD3(2), BRD2(2) and BRD4(2), respectively). |
Targets&IC50 | BRD2(2):830 nM (Kd), BRD3(2):490 nM (Kd), BRD4(2):850 nM (Kd), BRD4(1):160 nM (Kd), BRD3(1):380 nM (Kd), BRD2(1):170 nM (Kd) |
Molecular Weight | 421.51 |
Formula | C20H27N3O5S |
CAS No. | 1370888-71-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.21 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
XD14 1370888-71-3 Chromatin/Epigenetic Epigenetic Reader Domain XD 14 Inhibitor XD-14 inhibit inhibitor