20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12314 | Opioid receptor modulator 1 | Opioid Receptor | |
Opioid receptor modulator 1 is a modulator of opioid receptor. | |||
T62673 | Mu opioid receptor antagonist 5 | ||
Mu opioid receptor antagonist 5 (compound NAP) is a selective mu opioid receptor (MOR) antagonist that crosses the blood-brain barrier (EC50: 1.14 nM, Ki: 0.37 nM). Mu opioid receptor antagonist 5 can be used to study op... | |||
T62766 | Mu opioid receptor antagonist 2 | ||
Mu opioid receptor antagonist 2 (compound 25) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM). Mu opioid receptor antagonist 2 can be used... | |||
T62768 | Mu opioid receptor antagonist 4 | ||
Mu opioid receptor antagonist 4 (compound 31) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.38 nM, EC50: 0.38 nM). Mu opioid receptor antagonist 2 can be used... | |||
T79430 | μ opioid receptor agonist 3 | Opioid Receptor | |
Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM. It holds promise for research into pain management and neuropsychiatric disorders [1]. | |||
T62767 | Mu opioid receptor antagonist 3 | ||
Mu opioid receptor antagonist 3 (compound 26) is a potent and selective mu opioid receptor (MOR) antagonist that penetrates the blood-brain barrier (Ki: 0.24 nM, EC50: 0.54 nM). Mu opioid receptor antagonist 2 can be use... | |||
T62025 | μ opioid receptor agonist 2 | ||
μ opioid receptor agonist 2 (Compound H-3)is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases. | |||
T79431 | Mu opioid receptor antagonist 7 | Opioid Receptor | |
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (IC50) of 29 ± 3.0 nM. It is valuable for pain and opioid use ... | |||
T62268 | μ opioid receptor agonist 1 | ||
μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can be used in the study of pain and pain-related disorders. | |||
T61901 | σ1 Receptor/μ Opioid receptor modulator 1 | ||
σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM). Opioid receptor modulator 1 shows potent analgesic activity, and ... | |||
T6S1010 | Allomatrine | Others | |
Allomatrine is a natural product from Sophora alopecuroides L. Allomatrine, when given i.c.v., may stimulate the descending dynorphinergic neuron, resulting in the stimulation of KORs in the spinal cord. | |||
T7748 | Dermorphin TFA | Others , Opioid Receptor | |
Dermorphin TFA is a new class of opioids-like peptides | |||
T4691 | Asimadoline hydrochloride | EMD-61753 hydrochloride | Opioid Receptor |
Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also been shown to be used in the treatment of irritable bowel s... | |||
T9459 | GR103545 | Others | |
GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging. | |||
T4407 | SR17018 | Opioid Receptor | |
SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM. | |||
T4386 | PZM21 | Opioid Receptor | |
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM). | |||
T8992 | BMS986188 | Opioid Receptor | |
BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor. | |||
TP1832 | Gluten Exorphin C | Opioid Receptor | |
Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD assays, respectively.Gluten Exorphin C, isolated from the pe... | |||
T1242 | Alvimopan | Opioid Receptor | |
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvimopan is a selective and competitive antagonist at mu-opioid... | |||
T8991 | BMS986187 | Opioid Receptor | |
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor. |