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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15795 | Luzindole | N-0774 | Melatonin Receptor , MT Receptor |
Luzindole (N-0774) is a selective melatonin receptor antagonist. Luzindole inhibits experimental autoimmune encephalomyelitis and exerts antidepressant-like activity. Luzindole preferentially targets MT2 (Mel1b) over MT1... | |||
T23394 | SR 57227A | SR 57227 hydrochloride | 5-HT Receptor |
SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier. It has affinities (IC50) varying between 2.8 and 250 nM for 5-HT3 rece... | |||
T38007 | Noladin ether | ||
Noladin ether is a selective cannabinoid CB1 receptor agonist (Ki=21.2 nM). Noladin ether can cause hypothermia, intestinal immobility, and mild pain relief. | |||
T38109 | Galanin (2-11) amide (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt) | ||
Galanin (2-11) amide is a synthetic peptide fragment of the neuropeptide galanin and an agonist of the galanin-2 (GAL2) receptor (EC50= 9.32 nM in a fluorescence imaging plate reader assay).1It selectively binds to the G... | |||
T80693 | β-Endorphin, rat | β-Lipotropin 61-91 | |
β-Endorphin, rat (β-Lipotropin 61-91), a neuropeptide, plays a role in cardiovascular regulation and has been shown to cause significant, lasting muscular rigidity and immobility, akin to catatonia, in rats [1] [2]. | |||
T83676 | Tianeptine Metabolite MC5 sodium | ||
Tianeptine metabolite MC5, an active derivative of the atypical antidepressant tianeptine produced through β-oxidation, exhibits selective G protein activation in bioluminescence resonance energy transfer (BRET) assays. ... | |||
T83733 | TIP39 (human, bovine) TFA | Tuberoinfundibular Peptide of 39 Residues | |
TIP39, a neuropeptide and an agonist for the parathyroid hormone receptor type 2 (PTH2R), effectively increases cAMP levels in COS-7 cells featuring recombinant PTH2R from humans or rats (EC50s = 0.5 and 0.8 nM, respecti... | |||
T36521 | Alaproclate (hydrochloride) | ||
Alaproclate is a selective serotonin reuptake inhibitor (SSRI).1,2 It inhibits depletion of serotonin (5-HT) induced by 4-methyl-α-ethyl-m-tyramine in rat cerebral cortex, hippocampus, hypothalamus, and striatum (EC50s =... | |||
T37194 | 5α-Androst-16-en-3α-ol | ||
5α-Androst-16-en-3α-ol is a steroid pheromone that has been found in boar testes and human male axillary sweat and has diverse biological activities.1,2It enhances GABA-activated currents in primary mouse cerebellar gran... |