sigma-ligand-1 — TargetMol Chemicals

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Search Results for " sigma-ligand-1 "

Compounds

Cat No.	Product Name	Synonyms	Targets
T13510	Sigma-LIGAND-1		Sigma receptor
	Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively. Sigma-LIGAND-1 has a Ki of 4000 nM at the dopamine D2 receptor.		Sigma receptor
T63048	Sigma-LIGAND-1 hydrochloride
	Sigma-LIGAND-1 hydrochloride is a selective sigma receptor ligand that acts at the DTG (IC50: 16 nM) and PPP (IC50: 19 nM) sites. Sigma-LIGAND-1 hydrochloride is able to act on the dopamine D2 receptor (Ki: 4000 nM).
T39211	PD 144418 oxalate		Sigma receptor
	PD 144418 oxalate is a highly potent and selective sigma 1 (σ1) receptor ligand, displaying a Ki value of 0.08 nM for σ1 and 1377 nM for σ2. It exhibits negligible affinity for other receptors, ion channels, and enzymes....		Sigma receptor
T50090	3-(2-phenylethynyl)pyridine		Others
	3-(2-phenylethynyl)pyridine is a pyridine derivative that is a ligand for a variety of receptors in the human body, including dopamine D2 receptors, sigma-1 receptors, and 5-HT6 receptors. It has been studied for the tre...		Others
T25584	KSCM-1	KSCM 1
	KSCM-1 is a selective sigma-1 receptor ligand.
T26100	RLH 033	RLH033,RLH-033
	RLH 033 is a selective ligand for the sigma 1 recognition site.
T16445	PD 144418		Sigma receptor
	PD 144418 displays potential antipsychotic activity. PD 144418 is a high affinity, potent and selective sigma 1 (σ1) receptor ligand (Ki: 0.08 nM and 1377 nM for σ1 and σ2 respectively). It shows devoid of any significan...		Sigma receptor
T61846	CM398
	CM398 is an orally active chemical compound that acts as a highly selective ligand for the sigma-2 receptor (K i =0.43 nM), demonstrating a significant ratio of selectivity between sigma-1 and sigma-2 receptors (1000-fol...