3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13312L | Seviteronel | VT-464 | P450 , Androgen Receptor |
Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer. | |||
T13313 | Seviteronel racemate | VT-464 (racemate) | Others |
Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase. | |||
T13312 | Seviteronel R enantiomer | VT-464 (R enantiomer) | Others |
Seviteronel R enantiomer is the R enantiomer of Seviteronel and is a potent inhibitor of CYP17 lyase (IC50: 69 nM for h-Lyase). |