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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T61074 | Pim-1 kinase inhibitor 3 | ||
Pim-1 kinase inhibitor 3 (Compound H5) is a potent inhibitor of Pim-1 kinase, demonstrating an inhibitory concentration (IC50) of 35.13 nM [1]. | |||
T77526 | Pim-1 kinase inhibitor 4 | Apoptosis , Pim | |
Pim-1 kinase inhibitor 4 is a potent Pim-1 kinase inhibitor with an IC50 value of 17.01 nM.Pim-1 kinase inhibitor 4 also possesses antioxidant activity and potential anticancer activity, and inhibits DPPH.Pim-1 kinase in... | |||
T4523 | TP-3654 | Pim | |
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM). | |||
T6148 | CX-6258 hydrochloride | CX-6258 HCl,Pim-Kinase Inhibitor X | Pim |
CX-6258 hydrochloride (Pim-Kinase Inhibitor X) is an effective, orally efficacious Pim1/2/3 kinase inhibitor (IC50: 5/25/16 nM). | |||
T1834 | CX-6258 | CX 6258 | Pim |
CX-6258 is an orally valid Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor. It has good biological activity and kinase specificity. | |||
T3078 | SGI-1776 | SGI-1776 free base,Pim-Kinase Inhibitor IX | Apoptosis , FLT , Pim , Autophagy |
SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias. | |||
T63589 | CX-6258 hydrochloride hydrate | ||
CX-6258 hydrochloride hydrate is a potent and selective inhibitor of pan-Pim kinase that acts on Pim-1 (IC50: 5 nM), Pim-2 (IC50: 25 nM) and Pim-3 (IC50: 16 nM). |