pln — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T60101	PLN-1474	PLN1474	Integrin
	PLN-1474 is a potent αVβ1 inhibitor with IC50 < 50 nM.		Integrin
T39933	Bexotegrast	PLN-74809	Integrin
	Bexotegrast (PLN-74809) is an orally active and potent inhibitor of αvβ6 and αvβ1 integrins with antifibrotic effects, inhibits αvβ6 and αvβ1-induced activation of TGF-β, and can be used for the study of idiopathic pulmo...		Integrin
T69517	Bexotegrast HCl
	Bexotegrast, also known as PLN-74809, is a small-molecule, dual selective inhibitor of αVβ1 / αVβ6 for idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC). These integrins cause upstream activati...
T25492	Hepln-13	Hepln 13,Hepln13	c-Met/HGFR
	Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.		c-Met/HGFR
T35829	CC-90005
	CC-90005 is a potent, selective and orally active inhibitor of protein kinase C-θ (PKC-θ), with an IC50 of 8 nM. CC-90005 shows selectivity for PKC-θ over PKC-δ (IC50=4440 nM). CC-90005 can inhibit T cell activation by I...

Compounds

PLN-1474

T60101

Synonym: Hepln 13,Hepln13

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPH-01049	Cardiac phospholamban/PLN Protein, Human, Recombinant (GST)	Human	P. pastoris (Yeast)
	Cardiac phospholamban/PLN Protein, Human, Recombinant (GST) is expressed in yeast with N-GST tag. The predicted molecular weight is 33.1 kDa and the accession number is P26678.
TMPH-01504	HAPLN2 Protein, Human, Recombinant (His)	Human	E. coli
	Mediates a firm binding of versican V2 to hyaluronic acid. May play a pivotal role in the formation of the hyaluronan-associated matrix in the central nervous system (CNS) which facilitates neuronal conduction and genera...
TMPY-06365	APLN Protein, Mouse, Recombinant (mFc)	Mouse	HEK293 Cells
	APLN Protein, Mouse, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 33.57 kDa and the accession number is Q9R0R4.
TMPK-01222	APLN Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Macrophages play key roles during cardiovascular diseases (CVD) and their related complications.Apelin (APLN) is a key molecule, whose roles during CVD have been documented previously. Therefore, it has been hypothesized...
TMPH-02713	HAPLN3 Protein, Mouse, Recombinant (E. coli, His & Myc)	Mouse	E. coli
	HAPLN3 Protein, Mouse, Recombinant (E. coli, His & Myc) is expressed in E. coli.
TMPH-02714	HAPLN3 Protein, Mouse, Recombinant (His & Myc)	Mouse	HEK293 Cells
	May function in hyaluronic acid binding. HAPLN3 Protein, Mouse, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predicted molecular weight is 43.9 kDa and the accession num...
TMPY-00819	HAPLN1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Hyaluronan (HA) is a high MW glycosaminoglycan significantly involved in the formation and stability of extracellular matrix via its association with specific HA-binding proteins. HAPLN1, also known as CRTL1 (Cartilage L...
TMPH-01505	HAPLN3 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	May function in hyaluronic acid binding. HAPLN3 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with N-10xHis tag. The predicted molecular weight is 41.6 kDa and the accession number is Q96S86.
TMPH-01507	HAPLN4 Protein, Human, Recombinant (His)	Human	E. coli
	Binds to hyaluronic acid and may be involved in formation of the extracellular matrix.
TMPH-01506	HAPLN3 Protein, Human, Recombinant (E. coli, His)	Human	E. coli
	May function in hyaluronic acid binding. HAPLN3 Protein, Human, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 42.8 kDa and the accession number ...
TMPK-01236	APLN Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Macrophages play key roles during cardiovascular diseases (CVD) and their related complications.Apelin (APLN) is a key molecule, whose roles during CVD have been documented previously. Therefore, it has been hypothesized...
TMPK-01221	APLN Protein, Mouse, Recombinant (hFc & Avi), Biotinylated	Mouse	HEK293 Cells
	Macrophages play key roles during cardiovascular diseases (CVD) and their related complications.Apelin (APLN) is a key molecule, whose roles during CVD have been documented previously. Therefore, it has been hypothesized...