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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60452 | PCAF-IN-2 | ||
PCAF-IN-2 (compound 17) is a potent inhibitor of PCAF with an IC50 of 5.31 µM. PCAF-IN-2 exhibits anti-tumor activity. CAF-IN-2 induces cell apoptosis and arrest the cell cycle at the G2/M phase[1]. | |||
T5468 | YF-2 | Others , Epigenetic Reader Domain , Histone Acetyltransferase | |
YF-2 is blood-brain-barrier permeable histone acetyltransferase activator, acetylates H3 in the hippocampus, CBP, PCAF, and GCN5 with EC50s of 2.75 μM, 29.04 μM and 49.31 μM , respectively | |||
T35818 | CAY10669 | ||
CAY10669 is an inhibitor of the histone acetyltransferase PCAF (p300/CREB-binding protein-associated factor; IC50 = 662 μM), displaying a 2-fold improvement in inhibitory potency over anacardic acid . At 30-60 μM, CAY106... | |||
T38711 | YF-2 hydrochloride | ||
YF-2 hydrochloride is a potent histone acetyltransferase activator that exhibits high selectivity and can pass through the blood-brain barrier. It specifically acetylates H3 in the hippocampus, with EC50 values of 2.75 μ... |