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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2252 | UNC 669 | UNC669 | Epigenetic Reader Domain |
UNC 669 is an effective and specific MBT (malignant brain tumor) inhibitor with IC50 of 4.2/3.1 uM for L3MBTL1/3. | |||
T9221 | UNC926 hydrochloride | Epigenetic Reader Domain | |
UNC926 hydrochloride is a methyl-lysine (Kme) reader domain inhibitor. | |||
T4012 | UNC926 | UNC-926,UNC 926 hydrochloride | Epigenetic Reader Domain |
UNC926 (UNC-926) inhibits L3MBTL1 (IC50: 3.9 μM). UNC926 also exhibits a low micromolar affinity for L3MBTL3. UNC926 inhibits binding of the 3xMBT domain to H4K20me1. It selectively and dose-dependently inhibits the L3MB... |