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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1073 | Neuropeptide W-23(human) | NPW-23 | Others |
Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2. | |||
T62656 | GPR81 agonist 1 | GPR | |
GPR81 agonist 1 is a potent and selective GPR81 agonist with high affinity for human and mouse GPR81.GPR81 agonist 1 inhibits lipolysis of differentiated 3T3-L1 adipocytes, improves insulin sensitivity and glycaemic cont... | |||
T62261 | GPR84 antagonist 1 | ||
GPR84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human GPR84. | |||
T72536 | GPR84 antagonist 2 | ||
GPR84 Antagonist 2, a potent and selective GPR84 antagonist (IC 50 = 8.95 nM), demonstrates oral activity and significantly enhances potency in calcium mobilization assays. It effectively inhibits neutrophil and macropha... | |||
T11462 | GPR84 antagonist 8 | GPR | |
GPR84 antagonist 8 is a selective GPR84 antagonist. | |||
T72772 | GPR81 agonist 2 | ||
GPR81 agonist 2 is a potent agonist targeting the GPR81 receptor, demonstrating EC50 values of 0.023 µM for hGPR81 and 0.123 µM for hGPR109A, respectively. | |||
T62918 | GPR84 antagonist 3 | ||
GPR84 Antagonist 3 (compound 42), a potent inhibitor of the G-protein-coupled receptor 84 (GPR84), exhibits a pIC50 value of 8.28, indicating strong antagonistic activity by inhibiting GTPγS. Additionally, it possesses a... | |||
T79901 | GPR88-IN-1 | ||
GPR88-IN-1 is a GPR88 antagonist that may be utilized for the study of central nervous system disorders [1]. | |||
T79902 | GPR88 agonist 2 | ||
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1]. | |||
T81680 | Neuropeptide W-23 (human) (TFA) | NPW-23 TFA | |
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8) receptors [1]. | |||
T82862 | Biotinyl-neuropeptide W-23 (human) | ||
Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8) receptors [1] [2]. | |||
T83547 | (Des-Bromo)-Neuropeptide B (1-23) (human) | ||
'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM for GPR8 (NPBW2) respectively [1]. |