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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6484 | EI1 | KB-145943,Ezh2 inhibitor | Apoptosis , Histone Methyltransferase |
EI1 (Ezh2 inhibitor) is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively. | |||
T71871 | EI-1 | ||
EI-1 is an inhibitor of Hepatitis C virus entry. | |||
T9753 | LEI110 | Phospholipase | |
LEI110 is a potent Phospholipase A2, group XVI (PLA2G16) inhibitor with an Ki value of 20 nM. LEI110 is a selective pan-inhibitor of the HRASLS family of thiol hydrolases (i.e., PLA2G16, HRASLS2, RARRES3 and iNAT). | |||
T38377 | ADTL-EI1712 | ADTL-EI1712 | |
ADTL-EI1712 is a dual inhibitor of ERK1 and ERK5 (IC50s = 40.43 and 64.5 nM, respectively).1It reduces ERK1 and ERK5 activity by 93.5% and 89.4%, respectively, but also inhibits ERK2 activity by 92.7%, in a panel of 100 ... | |||
T27810 | LEI105 | LEI-105,LEI 105 | |
LEI105 is a potent, highly selective, and reversible inhibitor of DAGL-α and DAGL-β. |