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20

Compounds

Cat No. Product Name Synonyms Targets
TP1918L1 Lys-[Des-Arg9]Bradykinin acetate Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces p...
TP1918L Lys-[Des-Arg9]Bradykinin,TFA Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripher...
T1883 Des(benzylpyridyl) Atazanavi HIV Protease
The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.
T8809 [Des-Arg9]-Bradykinin TFA Bradykinin Receptor
[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
TP1445 [Des-Arg9]-Bradykinin acetate Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.
TP1917L1 Sar-[D-Phe8]-des-Arg9-Bradykinin acetate Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cl...
T1216 Diethylstilbestrol Stilbestrol,DES Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Diethylstilbestrol (DES) is used in the treatment of menopausal and postmenopausal disorders.
T7645 [Des-Arg9]-Bradykinin [Des-Arg9]-Bradykinin(2TFA) Bradykinin Receptor
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
TP1181 Bradykinin (2-9) Des-Arg1-bradykinin Bradykinin Receptor
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P.
TP2032 des-​Gln14-​Ghrelin des-Gln14-Ghrelin (rat)
An endogenous ligand for the ghrelin receptor (GHS-R1a), produced by alternative splicing of the rat ghrelin gene. Potently induces Ca2+ release in cells expressing ghrelin receptors (EC50 = 2.4 nM) and stimulates GH rel...
T36638 [Des-His1,Glu9]-Glucagon amide TFA [Des-His1,Glu9]-Glucagon amide TFA
[Des-His1,Glu9]-Glucagon amide TFA is a potent peptide antagonist targeting the glucagon receptor, featuring a pA2 value of 7.2. It holds potential utility in diabetes pathogenesis research[1].
T31634 [Des-Tyr1]-Met-Enkephalin Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-
Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats.
TP2033 [Des-His1,Glu9]-Glucagon amide des-His1-[Glu9]-Glucagon (1-29) amide
Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes); displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitr...
TP2450 Argipressin, des-glynh2(9)- 9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin
Argipressin, des-glynh2(9)-, can effect on aggregation of blood platelets.
TP1918 Lys-[Des-Arg9]Bradykinin
Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. ...
TP2241 [Des-octanoyl]-Ghrelin (human) Others
[Des-octanoyl]-Ghrelin (human) is a Non-acylated, major circulating isoform of ghrelin.
TP2242 [Des-octanoyl]-Ghrelin (rat) Others
[Des-octanoyl]-Ghrelin (rat) is a Non-acylated, major circulating isoform of ghrelin.
TP1917 Sar-[D-Phe8]-des-Arg9-Bradykinin
Potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic ac...
T35602 O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine
O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine is a major metabolite of the calcium channel inhibitor amlodipine .1 1.Taguchi, R., Naito, T., Sato, H., et al.Validated LC-MS/MS method for the simultaneous determin...
T83500 [Des-Arg10]-HOE I40
[Des-Arg10]-HOE 140 is a bioactive peptide that functions as a potent B1 bradykinin receptor antagonist.

Compounds

Lys-[Des-Arg9]Bradykinin acetate
TP1918L1
Synonym: Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA
TP1918L
Synonym: Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)
Target: Bradykinin Receptor
Des(benzylpyridyl) Atazanavi
T1883
Synonym:
Target: HIV Protease
[Des-Arg9]-Bradykinin TFA
T8809
Synonym:
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate
TP1445
Synonym:
Target: Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
TP1917L1
Synonym: Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)
Target: Bradykinin Receptor
Diethylstilbestrol
T1216
Synonym: Stilbestrol,DES
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
[Des-Arg9]-Bradykinin
T7645
Synonym: [Des-Arg9]-Bradykinin(2TFA)
Target: Bradykinin Receptor
Bradykinin (2-9)
TP1181
Synonym: Des-Arg1-bradykinin
Target: Bradykinin Receptor
des-​Gln14-​Ghrelin
TP2032
Synonym: des-Gln14-Ghrelin (rat)
Target:
[Des-His1,Glu9]-Glucagon amide TFA
T36638
Synonym: [Des-His1,Glu9]-Glucagon amide TFA
Target:
[Des-Tyr1]-Met-Enkephalin
T31634
Synonym: Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-
Target:
[Des-His1,Glu9]-Glucagon amide
TP2033
Synonym: des-His1-[Glu9]-Glucagon (1-29) amide
Target:
Argipressin, des-glynh2(9)-
TP2450
Synonym: 9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin
Target:
Lys-[Des-Arg9]Bradykinin
TP1918
Synonym:
Target:
[Des-octanoyl]-Ghrelin (human)
TP2241
Synonym:
Target: Others
[Des-octanoyl]-Ghrelin (rat)
TP2242
Synonym:
Target: Others
Sar-[D-Phe8]-des-Arg9-Bradykinin
TP1917
Synonym:
Target:
O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine
T35602
Synonym:
Target:
[Des-Arg10]-HOE I40
T83500
Synonym:
Target:
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TargetMol