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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1918L1 | Lys-[Des-Arg9]Bradykinin acetate | Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) | Bradykinin Receptor |
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces p... | |||
TP1918L | Lys-[Des-Arg9]Bradykinin,TFA | Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa) | Bradykinin Receptor |
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripher... | |||
T1883 | Des(benzylpyridyl) Atazanavi | HIV Protease | |
The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor. | |||
T8809 | [Des-Arg9]-Bradykinin TFA | Bradykinin Receptor | |
[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors. | |||
TP1445 | [Des-Arg9]-Bradykinin acetate | Bradykinin Receptor | |
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor. | |||
TP1917L1 | Sar-[D-Phe8]-des-Arg9-Bradykinin acetate | Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) | Bradykinin Receptor |
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cl... | |||
T1216 | Diethylstilbestrol | Stilbestrol,DES | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Diethylstilbestrol (DES) is used in the treatment of menopausal and postmenopausal disorders. | |||
T7645 | [Des-Arg9]-Bradykinin | [Des-Arg9]-Bradykinin(2TFA) | Bradykinin Receptor |
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor. | |||
TP1181 | Bradykinin (2-9) | Des-Arg1-bradykinin | Bradykinin Receptor |
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P. | |||
TP2032 | des-Gln14-Ghrelin | des-Gln14-Ghrelin (rat) | |
An endogenous ligand for the ghrelin receptor (GHS-R1a), produced by alternative splicing of the rat ghrelin gene. Potently induces Ca2+ release in cells expressing ghrelin receptors (EC50 = 2.4 nM) and stimulates GH rel... | |||
T36638 | [Des-His1,Glu9]-Glucagon amide TFA | [Des-His1,Glu9]-Glucagon amide TFA | |
[Des-His1,Glu9]-Glucagon amide TFA is a potent peptide antagonist targeting the glucagon receptor, featuring a pA2 value of 7.2. It holds potential utility in diabetes pathogenesis research[1]. | |||
T31634 | [Des-Tyr1]-Met-Enkephalin | Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)- | |
Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats. | |||
TP2033 | [Des-His1,Glu9]-Glucagon amide | des-His1-[Glu9]-Glucagon (1-29) amide | |
Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes); displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitr... | |||
TP2450 | Argipressin, des-glynh2(9)- | 9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin | |
Argipressin, des-glynh2(9)-, can effect on aggregation of blood platelets. | |||
TP1918 | Lys-[Des-Arg9]Bradykinin | ||
Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. ... | |||
TP2241 | [Des-octanoyl]-Ghrelin (human) | Others | |
[Des-octanoyl]-Ghrelin (human) is a Non-acylated, major circulating isoform of ghrelin. | |||
TP2242 | [Des-octanoyl]-Ghrelin (rat) | Others | |
[Des-octanoyl]-Ghrelin (rat) is a Non-acylated, major circulating isoform of ghrelin. | |||
TP1917 | Sar-[D-Phe8]-des-Arg9-Bradykinin | ||
Potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic ac... | |||
T35602 | O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine | ||
O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine is a major metabolite of the calcium channel inhibitor amlodipine .1 1.Taguchi, R., Naito, T., Sato, H., et al.Validated LC-MS/MS method for the simultaneous determin... | |||
T83500 | [Des-Arg10]-HOE I40 | ||
[Des-Arg10]-HOE 140 is a bioactive peptide that functions as a potent B1 bradykinin receptor antagonist. |