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Search Results for " bira "

Targets

13

Compounds

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T6216 Abiraterone CB-7598 P450
Abiraterone (CB-7598) (CB-7598) is an effective steroidal cytochrome P450 17alpha-hydroxylase-17, 20-lyase (CYP17) inhibitor (IC50: 4 nM).
T6032 Birabresib OTX-015,OTX015 (MK 8628/Birabresib),MK-8628 Epigenetic Reader Domain
Birabresib (MK-8628) is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4 with potential antineoplastic activity.
T6215 Abiraterone Acetate Zytiga,CB7630 P450
Abiraterone Acetate (CB7630) is an androstene derivative that inhibits STEROID 17-ALPHA-HYDROXYLASE and is used as an ANTINEOPLASTIC AGENT in the treatment of metastatic castration-resistant PROSTATE CANCER.
T74684 Abiraterone sulfate
Abiraterone sulfate is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .
TP2379 Ebiratide Ebiratida,Ebiratidum
Ebiratide is an analog of ACTH 4-9.
T74094 5,6-Dihydroabiraterone
5,6-Dihydroabiraterone, a metabolic derivative of Abiraterone, is a potent and irreversible inhibitor of CYP17A1, exhibiting antiandrogen and antitumor activities, particularly effective against castration-resistant pros...
T83214 Abiraterone sulfate N-oxide
Abiraterone sulfate N-oxide, a carboxylic acid and major metabolite of Abiraterone, is utilized in prostate cancer research [1] [2].
T74685 Abiraterone N-oxide
Abiraterone N-oxide is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .
T63434 Abiraterone decanoate
Abiraterone decanoate is a prodrug of Abiraterone that provides controlled release and long-lasting CYP17 inhibition of Abiraterone using intramuscular (IM) delivery.
T13525 Abiraterone metabolite 1 3β-OH-5α-Abi Others
Abiraterone Metabolite 1, a 5β-reduced derivative of abiraterone, acts by inhibiting CYP17A1, thereby blocking androgen synthesis and extending survival in prostate cancer patients.
T76786 Cabiralizumab
Cabiralizumab (FPA 008), an anti-CSF1R monoclonal antibody (MAb), promotes T cell infiltration and boosts antitumor immune responses. It also prevents osteoclast activation, thereby inhibiting bone destruction, and is ut...
T69963 Birabresib dihydrate
Birabresib dihydrate was initially developed by Mitsubishi Tanabe Pharma Corporation, but then was licensed by OncoEthix, privately held biotechnology company. OTX015 is a selective bromodomains: BRD2, BRD3, and BRD4 inh...
T10946 D4-abiraterone Abiraterone D4A metabolite,CB-7627,Δ4-Abiraterone Androgen Receptor
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abiraterone is also an antagonist of androgen receptor.

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-03650 BirA Protein, E. coli, Recombinant (His & MBP) E. coli E. coli
The enzyme BirA is a key reagent because of its ability to biotinylate proteins at a specific residue in a recognition sequence. This enzyme is used to biotinylate the C termini of membrane proteins, allowing these prote...
TargetMol