Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 68.00 | |
5 mg | In stock | $ 89.00 | |
10 mg | In stock | $ 142.00 | |
25 mg | In stock | $ 267.00 | |
50 mg | In stock | $ 445.00 | |
100 mg | In stock | $ 656.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 93.00 |
Description | SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively. |
Targets&IC50 | D3 receptor:8.0 (pKi), 5-HT1B:<5.2 (pKi), 5-HT1D:5.0 (pKi), D2 receptor:6.0 (pKi) |
Synonyms | SB-277011A |
Molecular Weight | 438.56 |
Formula | C28H30N4O |
CAS No. | 215803-78-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.39 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
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SB-277011 215803-78-4 GPCR/G Protein Neuroscience Dopamine Receptor SB-277011A SB 277011 SB277011 inhibitor inhibit