Powder: -20°C for 3 years
In solvent: -80°C for 2 years
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly reverses stress-induced anorexia but has no effect on food intake in free-feeding rats. Exhibits anxiolytic-like activity in vivo.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 237.00 | |
50 mg | In stock | $ 2,165.00 | |
100 mg | In stock | $ 3,259.00 |
Description | Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly reverses stress-induced anorexia but has no effect on food intake in free-feeding rats. Exhibits anxiolytic-like activity in vivo. |
Synonyms | MCL 0020 |
Molecular Weight | 609.731 |
Formula | C34H39N7O4 |
CAS No. | 475498-26-1 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
25% ethanol / water: 2 mg/mL
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
MCL0020 475498-26-1 GPCR/G Protein Neuroscience Melanocortin Receptor MCL 0020 inhibit COS-1 Inhibitor MC Receptor anorexia dose-dependently stress-induced MCL-0020 inhibitor