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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
NF-κB
Antibacterial
ROS
CDK
COX
PI3K
Dopamine Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Potassium Channel
AChR
EGFR
VEGFR
HIV Protease
Akt
Cytochromes P450
ERK
Reactive Oxygen Species
Calcium Channel
Antibiotic
p38 MAPK
TNF
Parasite
Ras
Histamine Receptor
mTOR
Caspase
Epigenetic Reader Domain
Sodium Channel
PPAR
JAK
Interleukin
Src
Virus Protease
NO Synthase
Ferroptosis
PDGFR
FLT
Estrogen/progestogen Receptor
iGluR
STAT
PDE
Dehydrogenase
Bcl-2 Family
SARS-CoV
HDAC
FGFR
IL Receptor
Influenza Virus
Wnt/beta-catenin
PKC
Histone Methyltransferase
Estrogen Receptor/ERR
TRP/TRPV Channel
c-Kit
PARP
JNK
GSK-3
GABA Receptor
AMPK
MMP
Antifungal
Microtubule Associated
NMDAR
c-Met/HGFR
Cholinesterase (ChE)
Prostaglandin Receptor
MDM-2/p53
Bcr-Abl
GluR
Raf
TLR
ALK
MAPK
HSV
Monoamine Oxidase
Phosphatase
MAO
TGF-beta/Smad
HIF/HIF Prolyl-Hydroxylase
Tyrosine Kinases
Mitophagy
Beta Amyloid
Aurora Kinase
Topoisomerase
Drug Metabolite
Proteasome
HSP
HCV Protease
MEK
GPCR
Casein Kinase
Lipoxygenase
PKA
P-gp
Nrf2
Serotonin Transporter
Norepinephrine
Cannabinoid Receptor
Reverse Transcriptase
ATPase
E1/E2/E3 Enzyme
p53
Sirtuin
Adenosine Receptor
IκB/IKK
Mitochondrial Metabolism
IGF-1R
ROCK
RAAS
S6 Kinase
LPL Receptor
Phospholipase
Antiviral
Anti-infection
NOS
Serine Protease
TAM Receptor
Gamma-secretase
HBV
Glucocorticoid Receptor
Trk receptor
S1P Receptor
DNA-PK
Serine/threonin kinase
Opioid Receptor
Retinoid Receptor
HIF
Carbonic Anhydrase
Nucleoside Antimetabolite/Analog
HER
c-RET
NOD-like Receptor (NLR)
Antioxidant
Integrin
DUB
Androgen Receptor
Cysteine Protease
Tyrosinase
Histone Acetyltransferase
FAK
c-Fms
CaMK
PROTACs
Progesterone Receptor
Histone Demethylase
PERK
Mdm2
Transferase
Pim
CXCR
DYRK
NOD
Angiotensin-converting Enzyme (ACE)
CCR
Hedgehog/Smoothened
ATM/ATR
DNA Alkylator/Crosslinker
Rho
ROS Kinase
HMG-CoA Reductase
Syk
Reductase
Glucosidase
Glutathione Peroxidase
RIP kinase
Immunology/Inflammation related
Chk
PLK
Sigma receptor
Beta-Secretase
BACE
NADPH
transporter
DNA Methyltransferase
Aryl Hydrocarbon Receptor
MRP
Kras
DPP-4
Antifection
Fatty Acid Synthase
Smo
IDO
Proton pump
P2X Receptor
Indoleamine 2,3-Dioxygenase (IDO)
FAAH
Acyltransferase
AhR
Chloride channel
c-Myc
PAK
glycosidase
DNA
DNA Alkylation
Leukotriene Receptor
GPCR19
IAP
CSF-1R
Stearoyl-CoA Desaturase (SCD)
SGLT
PDK
Isocitrate Dehydrogenase (IDH)
Kinesin
LTR
ABC Transporter
ADC Cytotoxin
YAP
Thrombin
FXR
Liver X Receptor
cAMP
IRAK
P2Y Receptor
Melatonin Receptor
LDL
PGE Synthase
Amino Acids and Derivatives
MNK
Tie-2
IFNAR
Telomerase
Lipid
LPA Receptor
PTEN
Pyroptosis
PD-1/PD-L1
UGT
Discoidin Domain Receptor (DDR)
PI4K
CFTR
DHFR
Myosin
Endothelin Receptor
Necroptosis
MT Receptor
Molecular Glues
OXPHOS
LRRK2
OX Receptor
BCRP
BTK
LIM Kinase
Monoamine Transporter
ribosome
DNA gyrase
Xanthine Oxidase
Epoxide Hydrolase
MLK
GTPase
Aromatase
Antifolate
PYK2
MicroRNA
ROR
Ligands for Target Protein for PROTAC
Lipase
PAFR
RSV
Thyroid hormone receptor(THR)
Annexin A
SGK
STING
Free radical scavengers
NADPH-oxidase
Vasopressin Receptor
Ephrin Receptor
GST
Aminopeptidase
Glucagon Receptor
Complement System
Hydroxylase
SIK
Neurokinin receptor
Guanylate cyclase
FKBP
Arginase
PAI-1
Platelet aggregation
Adenylate cyclase
Survivin
IKZF
Glucokinase
OAT
ATP Citrate Lyase
CRISPR/Cas9
Imidazoline Receptor
Phosphorylase
RAR/RXR
MyD88
Arrestin
IRE1
MAGL
Cadherin
GPX
Factor Xa
NAMPT
Glutaminase
ASK
Protease-activated Receptor
Dynamin
MTH1
NR4A
Porcupine
cGAS
NPC1L1
AAK1
Decarboxylase
FOXO
Bcl-6
GRK
ACK1
Na+/Ca2+ Exchanger
AIM2
Carboxypeptidase
Hexokinase
NEDD8
ATG
Melanin-concentrating Hormone Receptor (MCHR)
TOPK
Cholecystokinin Receptor
Adenosine Deaminase
OCT
Hck
RANKL/RANK
Bombesin Receptor
Amylase
GluCls
CGRP Receptor
CRFR
Melanocortin Receptor
GHSR
Gap Junction Protein
Transaminase
GlyT
Ligands for E3 Ligase
PAD
Thrombopoietin Receptor
Wee1
Methionine Adenosyltransferase (MAT)
Aquaporin
Cuproptosis
FOXO3
Cell Cycle Arrest
Haspin Kinase
Orphan Receptor
Protease
KLF
VDA
Adiponectin Receptor
PROTAC Linker
Hippo pathway
p62
LDLR
FLAP
Neuropeptide FF Receptor
Glutathione reductase
Neprilysin
Advanced Glycation End Products
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
Na-K-Cl cotransporter
BMI-1
Monocarboxylate transporter
FABP
KSP
Huntingtin
PKM
gp120/CD4
GNRH Receptor
ASCT
CPT
MELK
Oxytocin Receptor
REV-ERB
Lysosomal Autophagy
CRM1
MIF
DAPK
Tight Junction Protein
N-Acetylglucosaminyltransferase
Anion Exchanger
CD74
Taste receptor
Aconitase
Integrase
APC/C
Cell wall
CETP
Fas/FasL
Neuropeptide Y Receptor
hCE
Prolyl Endopeptidase (PREP)
Acetyl-CoA Carboxylase
RXFP receptor
ATTECs
CAT
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
CaSR
Photosensitizer
HCN Channel
Somatostatin
Urea Transporter
p97

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