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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
NF-κB
CDK
Dopamine Receptor
COX
PI3K
Antibacterial
Adrenergic Receptor
AChR
EGFR
Potassium Channel
HIV Protease
DNA/RNA Synthesis
VEGFR
Cytochromes P450
Calcium Channel
Histamine Receptor
Antibiotic
Reactive Oxygen Species
Akt
TNF
Epigenetic Reader Domain
ERK
Sodium Channel
mTOR
JAK
Estrogen/progestogen Receptor
Src
PPAR
PDGFR
FLT
PDE
p38 MAPK
Dehydrogenase
Parasite
IL Receptor
Ferroptosis
HDAC
FGFR
Histone Methyltransferase
PKC
iGluR
Influenza Virus
STAT
c-Kit
TRP/TRPV Channel
Wnt/beta-catenin
Caspase
SARS-CoV
Estrogen Receptor/ERR
PARP
GABA Receptor
Bcl-2 Family
AMPK
GSK-3
NMDAR
Microtubule Associated
NO Synthase
ALK
c-Met/HGFR
MMP
GluR
Antifungal
MAO
Bcr-Abl
ROS
Raf
Tyrosine Kinases
Virus Protease
Cholinesterase (ChE)
Aurora Kinase
MAPK
Prostaglandin Receptor
Mitophagy
Topoisomerase
TLR
HSV
Ras
JNK
Phosphatase
Proteasome
Beta Amyloid
HCV Protease
TGF-beta/Smad
HIF/HIF Prolyl-Hydroxylase
Lipoxygenase
HSP
ATPase
MEK
GPCR
PKA
Norepinephrine
Casein Kinase
p53
Interleukin
Cannabinoid Receptor
Adenosine Receptor
Mitochondrial Metabolism
Sirtuin
Reverse Transcriptase
ROCK
Monoamine Oxidase
E1/E2/E3 Enzyme
Antiviral
Nrf2
NOS
RAAS
IκB/IKK
TAM Receptor
LPL Receptor
Serotonin Transporter
Drug Metabolite
IGF-1R
P-gp
Phospholipase
S6 Kinase
Glucocorticoid Receptor
DNA-PK
Serine/threonin kinase
Retinoid Receptor
HIF
S1P Receptor
HER
Carbonic Anhydrase
Antioxidant
Gamma-secretase
Trk receptor
c-RET
HBV
DUB
Opioid Receptor
Integrin
Nucleoside Antimetabolite/Analog
Androgen Receptor
Progesterone Receptor
Serine Protease
Mdm2
Histone Demethylase
Cysteine Protease
Tyrosinase
Pim
Rho
Histone Acetyltransferase
c-Fms
NOD
PERK
CCR
CXCR
CaMK
HMG-CoA Reductase
FAK
PROTACs
Transferase
DNA Alkylator/Crosslinker
BACE
DYRK
Hedgehog/Smoothened
ATM/ATR
Syk
MRP
PLK
DNA Methyltransferase
Sigma receptor
DPP-4
Chk
transporter
NADPH
Aryl Hydrocarbon Receptor
RIP kinase
P2X Receptor
Smo
NOD-like Receptor (NLR)
Chloride channel
Glutathione Peroxidase
Glucosidase
Fatty Acid Synthase
Acyltransferase
AhR
Proton pump
Immunology/Inflammation related
DNA Alkylation
FAAH
DNA
Indoleamine 2,3-Dioxygenase (IDO)
Beta-Secretase
CSF-1R
PAK
cAMP
PDK
ROS Kinase
LTR
Reductase
IAP
LDL
ABC Transporter
Antifection
Stearoyl-CoA Desaturase (SCD)
Thrombin
Kinesin
P2Y Receptor
SGLT
GPCR19
IRAK
ADC Cytotoxin
YAP
c-Myc
Liver X Receptor
Isocitrate Dehydrogenase (IDH)
PGE Synthase
MNK
LPA Receptor
DHFR
Leukotriene Receptor
FXR
IDO
UGT
MT Receptor
Endothelin Receptor
LRRK2
IFNAR
GTPase
Melatonin Receptor
Antifolate
Myosin
DNA gyrase
BTK
OX Receptor
Xanthine Oxidase
Epoxide Hydrolase
Lipid
ribosome
Aromatase
PI4K
Discoidin Domain Receptor (DDR)
CFTR
Thyroid hormone receptor(THR)
ROR
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
LIM Kinase
PYK2
Monoamine Transporter
Vasopressin Receptor
Telomerase
BCRP
STING
Free radical scavengers
Ephrin Receptor
GST
SGK
Anti-infection
NADPH-oxidase
MLK
PD-1/PD-L1
MicroRNA
Arginase
Lipase
Tie-2
SIK
PAFR
Guanylate cyclase
PTEN
Aminopeptidase
CRISPR/Cas9
Neurokinin receptor
Platelet aggregation
IKZF
Factor Xa
Glucokinase
NAMPT
Annexin A
Glucagon Receptor
Phosphorylase
ASK
RSV
GPX
Complement System
Protease-activated Receptor
Imidazoline Receptor
NPC1L1
RAR/RXR
Dynamin
MyD88
Na+/Ca2+ Exchanger
Arrestin
Bcl-6
AAK1
IRE1
MTH1
GRK
ACK1
ATP Citrate Lyase
OAT
Porcupine
Decarboxylase
PAI-1
Pyroptosis
Carboxypeptidase
Hydroxylase
Kras
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
Transaminase
NEDD8
TOPK
Cholecystokinin Receptor
Hck
Glutaminase
Amylase
GlyT
Hexokinase
Molecular Glues
MAGL
PAD
Thrombopoietin Receptor
AIM2
cGAS
GluCls
Ligand for E3 Ligase
Melanocortin Receptor
GHSR
Adenosine Deaminase
Gap Junction Protein
FOXO3
Advanced Glycation End Products
Monocarboxylate transporter
CRM1
gp120/CD4
VDA
OCT
GNRH Receptor
Cell Cycle Arrest
LDLR
FLAP
Neuropeptide FF Receptor
Adiponectin Receptor
Haspin Kinase
Bombesin Receptor
KSP
Cadherin
Orphan Receptor
Wee1
OXPHOS
Huntingtin
Glutathione reductase
CPT
CRFR
MELK
Neprilysin
Hippo pathway
Protease
KLF
Oxytocin Receptor
CGRP Receptor
DAPK
BMI-1
Lysosomal Autophagy
PKM
Taste receptor
GSNOR
EBI2/GPR183
Aconitase
Cell wall
CETP
Necroptosis
MIF
N-Acetylglucosaminyltransferase
CaSR
ASCT
Photosensitizer
ATG
NR4A
RANKL/RANK
Fas/FasL
FABP
Na-K-Cl cotransporter
Anion Exchanger
Integrase
PROTAC Linker
HCN Channel
Neuropeptide Y Receptor
Angiotensin-converting Enzyme (ACE)
Somatostatin
Survivin
Urea Transporter
hCE
Methionine Adenosyltransferase (MAT)
Acetyl-CoA Carboxylase
Aquaporin
FOXO
RXFP receptor
ATTECs
APC/C
p97

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