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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
NF-κB
CDK
Dopamine Receptor
COX
PI3K
Antibacterial
Adrenergic Receptor
AChR
EGFR
Potassium Channel
HIV Protease
DNA/RNA Synthesis
VEGFR
Cytochromes P450
Calcium Channel
Histamine Receptor
Antibiotic
Reactive Oxygen Species
Akt
TNF
Epigenetic Reader Domain
ERK
Sodium Channel
mTOR
JAK
Estrogen/progestogen Receptor
Src
FLT
PDGFR
PDE
PPAR
Dehydrogenase
p38 MAPK
IL Receptor
HDAC
Ferroptosis
FGFR
Parasite
Histone Methyltransferase
PKC
iGluR
STAT
c-Kit
Influenza Virus
TRP/TRPV Channel
Wnt/beta-catenin
SARS-CoV
Caspase
Estrogen Receptor/ERR
PARP
GABA Receptor
Bcl-2 Family
AMPK
NO Synthase
GSK-3
NMDAR
Microtubule Associated
ALK
MMP
GluR
c-Met/HGFR
ROS
MAO
Bcr-Abl
Raf
Antifungal
Virus Protease
Prostaglandin Receptor
MAPK
Cholinesterase (ChE)
Aurora Kinase
Mitophagy
Tyrosine Kinases
Topoisomerase
TLR
Ras
HSV
JNK
Phosphatase
Proteasome
Beta Amyloid
HCV Protease
HIF/HIF Prolyl-Hydroxylase
TGF-beta/Smad
Lipoxygenase
HSP
MEK
ATPase
Norepinephrine
p53
Cannabinoid Receptor
GPCR
PKA
Casein Kinase
Adenosine Receptor
Interleukin
Mitochondrial Metabolism
Sirtuin
ROCK
Monoamine Oxidase
Reverse Transcriptase
Nrf2
E1/E2/E3 Enzyme
Antiviral
RAAS
TAM Receptor
NOS
IκB/IKK
S6 Kinase
Drug Metabolite
LPL Receptor
Phospholipase
P-gp
Serotonin Transporter
IGF-1R
Glucocorticoid Receptor
Retinoid Receptor
Serine/threonin kinase
HIF
S1P Receptor
DNA-PK
HER
c-RET
Carbonic Anhydrase
Gamma-secretase
Antioxidant
DUB
Trk receptor
HBV
Opioid Receptor
Integrin
Androgen Receptor
Nucleoside Antimetabolite/Analog
Serine Protease
Progesterone Receptor
Histone Demethylase
Mdm2
Cysteine Protease
Tyrosinase
Pim
NOD
c-Fms
Rho
Histone Acetyltransferase
PERK
CCR
CXCR
HMG-CoA Reductase
FAK
Syk
Hedgehog/Smoothened
BACE
ATM/ATR
DNA Alkylator/Crosslinker
DYRK
CaMK
Transferase
PROTACs
Sigma receptor
PLK
MRP
DNA Methyltransferase
DPP-4
transporter
Chk
P2X Receptor
NADPH
RIP kinase
NOD-like Receptor (NLR)
Smo
Aryl Hydrocarbon Receptor
Glucosidase
Chloride channel
AhR
Glutathione Peroxidase
Fatty Acid Synthase
Acyltransferase
Indoleamine 2,3-Dioxygenase (IDO)
Beta-Secretase
Proton pump
Immunology/Inflammation related
FAAH
DNA
DNA Alkylation
CSF-1R
cAMP
PDK
ROS Kinase
PAK
Antifection
Stearoyl-CoA Desaturase (SCD)
LDL
IAP
Reductase
LTR
Thrombin
Kinesin
ABC Transporter
SGLT
IRAK
GPCR19
P2Y Receptor
ADC Cytotoxin
YAP
c-Myc
LPA Receptor
MNK
Liver X Receptor
PGE Synthase
Isocitrate Dehydrogenase (IDH)
IDO
Endothelin Receptor
Leukotriene Receptor
MT Receptor
DHFR
FXR
UGT
LRRK2
Discoidin Domain Receptor (DDR)
CFTR
Aromatase
Xanthine Oxidase
GTPase
PI4K
Melatonin Receptor
Lipid
OX Receptor
Myosin
DNA gyrase
Antifolate
IFNAR
ribosome
BTK
Amino Acids and Derivatives
GST
Thyroid hormone receptor(THR)
NADPH-oxidase
Monoamine Transporter
BCRP
Vasopressin Receptor
ROR
Ligands for Target Protein for PROTAC
Telomerase
PYK2
Free radical scavengers
Anti-infection
LIM Kinase
Epoxide Hydrolase
Ephrin Receptor
STING
PD-1/PD-L1
SGK
MLK
Aminopeptidase
Arginase
SIK
Lipase
Tie-2
PAFR
Platelet aggregation
CRISPR/Cas9
Guanylate cyclase
PTEN
MicroRNA
Glucokinase
ASK
Imidazoline Receptor
Factor Xa
RSV
Annexin A
Neurokinin receptor
Phosphorylase
Complement System
Protease-activated Receptor
GPX
NAMPT
Glucagon Receptor
NPC1L1
GRK
ACK1
Carboxypeptidase
Dynamin
IRE1
MyD88
Porcupine
Pyroptosis
RAR/RXR
Decarboxylase
MTH1
AAK1
OAT
ATP Citrate Lyase
Hydroxylase
PAI-1
Arrestin
Na+/Ca2+ Exchanger
Kras
Neuropeptide Y Receptor
TOPK
AIM2
Molecular Glues
Transaminase
Thrombopoietin Receptor
NEDD8
Cholecystokinin Receptor
Ligand for E3 Ligase
Hexokinase
MAGL
Adenosine Deaminase
Amylase
cGAS
GHSR
Glutaminase
GlyT
Adenylyl Cyclase
Melanin-concentrating Hormone Receptor (MCHR)
GluCls
Gap Junction Protein
Hck
PAD
Melanocortin Receptor
FOXO3
FLAP
Neprilysin
Huntingtin
Bombesin Receptor
Cell Cycle Arrest
KSP
PKM
CRM1
Wee1
Haspin Kinase
Protease
Glutathione reductase
OCT
DAPK
BMI-1
Hippo pathway
MELK
Adiponectin Receptor
Advanced Glycation End Products
Monocarboxylate transporter
OXPHOS
VDA
Lysosomal Autophagy
CRFR
KLF
CGRP Receptor
gp120/CD4
CPT
Oxytocin Receptor
GNRH Receptor
IKZF
Anion Exchanger
Integrase
Cell wall
N-Acetylglucosaminyltransferase
Methionine Adenosyltransferase (MAT)
Necroptosis
Na-K-Cl cotransporter
GSNOR
Aconitase
Somatostatin
APC/C
ATTECs
Acetyl-CoA Carboxylase
Survivin
Aquaporin
EBI2/GPR183
RXFP receptor
Fas/FasL
Taste receptor
CaSR
CETP
RANKL/RANK
PROTAC Linker
hCE
p97
FABP
HCN Channel
Angiotensin-converting Enzyme (ACE)

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