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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
NF-κB
CDK
Dopamine Receptor
COX
PI3K
Adrenergic Receptor
AChR
Potassium Channel
DNA/RNA Synthesis
EGFR
VEGFR
HIV Protease
Cytochromes P450
Reactive Oxygen Species
Calcium Channel
Antibiotic
Akt
Parasite
ERK
TNF
Ras
Histamine Receptor
Epigenetic Reader Domain
p38 MAPK
mTOR
Sodium Channel
PPAR
Src
JAK
Estrogen/progestogen Receptor
Virus Protease
PDGFR
FLT
Caspase
PDE
Dehydrogenase
Ferroptosis
iGluR
FGFR
HDAC
IL Receptor
Bcl-2 Family
Influenza Virus
SARS-CoV
STAT
PKC
Estrogen Receptor/ERR
Histone Methyltransferase
TRP/TRPV Channel
c-Kit
NO Synthase
Wnt/beta-catenin
PARP
Interleukin
GABA Receptor
GSK-3
AMPK
Microtubule Associated
MMP
Antifungal
c-Met/HGFR
NMDAR
GluR
MDM-2/p53
Bcr-Abl
Cholinesterase (ChE)
ALK
Raf
Prostaglandin Receptor
MAO
MAPK
Mitophagy
ROS
Monoamine Oxidase
Phosphatase
Tyrosine Kinases
HSV
Aurora Kinase
JNK
Topoisomerase
TGF-beta/Smad
TLR
Beta Amyloid
HIF/HIF Prolyl-Hydroxylase
HCV Protease
Proteasome
HSP
GPCR
Casein Kinase
MEK
Drug Metabolite
Lipoxygenase
ATPase
PKA
Reverse Transcriptase
Cannabinoid Receptor
Serotonin Transporter
Norepinephrine
p53
E1/E2/E3 Enzyme
Adenosine Receptor
Mitochondrial Metabolism
P-gp
Sirtuin
IκB/IKK
ROCK
Nrf2
LPL Receptor
S6 Kinase
IGF-1R
Antiviral
Phospholipase
Anti-infection
NOS
RAAS
TAM Receptor
Serine Protease
Glucocorticoid Receptor
DNA-PK
HBV
Gamma-secretase
Serine/threonin kinase
Retinoid Receptor
HIF
S1P Receptor
Carbonic Anhydrase
Nucleoside Antimetabolite/Analog
c-RET
HER
Antioxidant
Trk receptor
Opioid Receptor
DUB
Integrin
Androgen Receptor
Histone Acetyltransferase
c-Fms
Tyrosinase
NOD-like Receptor (NLR)
Progesterone Receptor
Cysteine Protease
FAK
Mdm2
Histone Demethylase
Pim
Transferase
DYRK
PERK
CXCR
NOD
DNA Alkylator/Crosslinker
Rho
CCR
CaMK
HMG-CoA Reductase
ROS Kinase
PROTACs
Glucosidase
Hedgehog/Smoothened
ATM/ATR
Syk
BACE
NADPH
MRP
Aryl Hydrocarbon Receptor
Beta-Secretase
PLK
DNA Methyltransferase
Sigma receptor
Kras
Glutathione Peroxidase
DPP-4
Angiotensin-converting Enzyme (ACE)
Chk
transporter
IDO
Immunology/Inflammation related
RIP kinase
P2X Receptor
Antifection
Smo
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Chloride channel
Proton pump
PAK
FAAH
Acyltransferase
AhR
c-Myc
DNA Alkylation
DNA
Reductase
Leukotriene Receptor
CSF-1R
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
cAMP
PDK
ADC Cytotoxin
LTR
FXR
IAP
LDL
ABC Transporter
SGLT
GPCR19
Thrombin
Kinesin
YAP
P2Y Receptor
Liver X Receptor
PGE Synthase
IRAK
IFNAR
Tie-2
Melatonin Receptor
UGT
Telomerase
MNK
Pyroptosis
LPA Receptor
DHFR
Amino Acids and Derivatives
Myosin
Endothelin Receptor
PTEN
OX Receptor
Lipid
OXPHOS
LRRK2
PI4K
Discoidin Domain Receptor (DDR)
CFTR
PD-1/PD-L1
BTK
GTPase
Antifolate
PYK2
MT Receptor
DNA gyrase
Monoamine Transporter
Molecular Glues
Xanthine Oxidase
Epoxide Hydrolase
BCRP
ribosome
Aromatase
Thyroid hormone receptor(THR)
MicroRNA
ROR
Ligands for Target Protein for PROTAC
LIM Kinase
Annexin A
Vasopressin Receptor
STING
Free radical scavengers
Aminopeptidase
Ephrin Receptor
RSV
GST
SGK
NADPH-oxidase
MLK
Arginase
Lipase
SIK
PAFR
Guanylate cyclase
PAI-1
FKBP
CRISPR/Cas9
Hydroxylase
Complement System
Neurokinin receptor
Platelet aggregation
IKZF
Arrestin
Necroptosis
Factor Xa
Glucokinase
NAMPT
Glucagon Receptor
Phosphorylase
MAGL
ATP Citrate Lyase
OAT
ASK
GPX
Protease-activated Receptor
Imidazoline Receptor
NPC1L1
RAR/RXR
Dynamin
MyD88
Na+/Ca2+ Exchanger
Bcl-6
AAK1
Glutaminase
NR4A
IRE1
MTH1
GRK
ACK1
Survivin
Porcupine
AIM2
Decarboxylase
cGAS
Carboxypeptidase
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
Transaminase
NEDD8
TOPK
OCT
Cholecystokinin Receptor
Hck
ATG
Amylase
GlyT
Hexokinase
Bombesin Receptor
PAD
Thrombopoietin Receptor
GluCls
CRFR
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Melanocortin Receptor
GHSR
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Gap Junction Protein
FOXO3
Advanced Glycation End Products
Monocarboxylate transporter
CRM1
gp120/CD4
MIF
VDA
GNRH Receptor
ASCT
Cell Cycle Arrest
LDLR
FLAP
Neuropeptide FF Receptor
Adiponectin Receptor
Haspin Kinase
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
Na-K-Cl cotransporter
KSP
Cadherin
Orphan Receptor
Wee1
Huntingtin
Glutathione reductase
CPT
MELK
Neprilysin
Hippo pathway
p62
Protease
KLF
Oxytocin Receptor
Aquaporin
FOXO
REV-ERB
DAPK
BMI-1
Lysosomal Autophagy
PKM
Taste receptor
CAT
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
Aconitase
Cell wall
CETP
N-Acetylglucosaminyltransferase
CaSR
Photosensitizer
RANKL/RANK
Prolyl Endopeptidase (PREP)
Fas/FasL
FABP
Anion Exchanger
Integrase
PROTAC Linker
HCN Channel
Neuropeptide Y Receptor
Somatostatin
Urea Transporter
hCE
Acetyl-CoA Carboxylase
RXFP receptor
ATTECs
APC/C
p97

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