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TargetMol | Compound Library

Multi-Target Compound Library

Catalog No. L9510

The pathogenesis of complex diseases often involves the interplay of multiple biological targets and signaling pathways, making it difficult for single-target drugs to achieve optimal therapeutic outcomes. As a result, single-target treatment strategies may have limited efficacy in certain cases. In contrast, multi-target drugs can act on multiple key targets or related pathways simultaneously, producing synergistic effects that significantly enhance therapeutic effectiveness.
This integrated intervention approach not only facilitates more comprehensive regulation of disease-associated biological networks but also helps to reduce the risk of drug resistance caused by mutations in individual targets. Moreover, due to the synergistic interactions between different targets, multi-target drugs can achieve desired therapeutic outcomes at lower dosages, thereby reducing toxicity and improving both safety and tolerability.
Therefore, multi-target drugs offer a more systematic and efficient strategy for the treatment of complex diseases.
TargetMol’s Multi-Target Compound Library contains 5200 compounds that act on two or more distinct targets, providing a valuable resource for the development of multi-target therapeutics.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9510

Multi-Target Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 5200 types of multi-target compounds for high throughput screening (HTS) and high content screening (HCS);
  • Approved by FDA and already on the market;
  • Structurally diverse, medicin active, and cell-permeable.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are available in stock for immediate delivery.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
NF-κB
CDK
ROS
PI3K
COX
Dopamine Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Potassium Channel
AChR
EGFR
VEGFR
HIV Protease
Cytochromes P450
Akt
Reactive Oxygen Species
Calcium Channel
ERK
Antibiotic
p38 MAPK
TNF
Parasite
Ras
Caspase
Histamine Receptor
mTOR
Epigenetic Reader Domain
PPAR
Sodium Channel
Src
JAK
Interleukin
NO Synthase
Ferroptosis
Virus Protease
Estrogen/progestogen Receptor
PDGFR
FLT
iGluR
PDE
Dehydrogenase
STAT
Bcl-2 Family
SARS-CoV
HDAC
FGFR
Influenza Virus
IL Receptor
Wnt/beta-catenin
PKC
Histone Methyltransferase
Estrogen Receptor/ERR
TRP/TRPV Channel
PARP
c-Kit
JNK
GSK-3
AMPK
GABA Receptor
Antifungal
MMP
Microtubule Associated
c-Met/HGFR
NMDAR
Prostaglandin Receptor
Bcr-Abl
MDM-2/p53
Cholinesterase (ChE)
GluR
TLR
Raf
ALK
HSV
MAPK
Phosphatase
MAO
Monoamine Oxidase
TGF-beta/Smad
Mitophagy
Tyrosine Kinases
Beta Amyloid
HIF/HIF Prolyl-Hydroxylase
Aurora Kinase
Topoisomerase
Drug Metabolite
Proteasome
HSP
HCV Protease
GPCR
MEK
PKA
Lipoxygenase
Nrf2
Casein Kinase
Norepinephrine
P-gp
Reverse Transcriptase
Cannabinoid Receptor
Serotonin Transporter
E1/E2/E3 Enzyme
p53
ATPase
Adenosine Receptor
Sirtuin
Mitochondrial Metabolism
IκB/IKK
ROCK
IGF-1R
LPL Receptor
S6 Kinase
NOS
RAAS
Antiviral
Phospholipase
Serine Protease
Anti-infection
TAM Receptor
HBV
Glucocorticoid Receptor
DNA-PK
Serine/threonin kinase
Gamma-secretase
Opioid Receptor
Trk receptor
Retinoid Receptor
HIF
S1P Receptor
Carbonic Anhydrase
PERK
Nucleoside Antimetabolite/Analog
c-RET
NOD-like Receptor (NLR)
HER
Integrin
Antioxidant
DUB
Androgen Receptor
Cysteine Protease
Histone Acetyltransferase
Tyrosinase
FAK
CaMK
c-Fms
Histone Demethylase
Progesterone Receptor
Mdm2
PROTACs
Pim
Transferase
DYRK
CXCR
NOD
HMG-CoA Reductase
DNA Alkylator/Crosslinker
Rho
Hedgehog/Smoothened
CCR
ATM/ATR
ROS Kinase
Reductase
Glutathione Peroxidase
RIP kinase
Glucosidase
Angiotensin-converting Enzyme (ACE)
transporter
Syk
BACE
NADPH
MRP
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
Chk
Beta-Secretase
PLK
DNA Methyltransferase
Sigma receptor
Kras
Antifection
DPP-4
Fatty Acid Synthase
Proton pump
IDO
P2X Receptor
Smo
Indoleamine 2,3-Dioxygenase (IDO)
Chloride channel
c-Myc
PAK
FAAH
Acyltransferase
AhR
Leukotriene Receptor
DNA Alkylation
glycosidase
DNA
CSF-1R
IAP
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
cAMP
SGLT
GPCR19
PDK
Kinesin
ADC Cytotoxin
YAP
LTR
Liver X Receptor
FXR
LDL
ABC Transporter
IRAK
Thrombin
P2Y Receptor
Melatonin Receptor
PGE Synthase
Amino Acids and Derivatives
IFNAR
Tie-2
UGT
PTEN
Telomerase
Lipid
MNK
Pyroptosis
LPA Receptor
Discoidin Domain Receptor (DDR)
PD-1/PD-L1
DHFR
Necroptosis
Myosin
MT Receptor
Molecular Glues
Endothelin Receptor
OX Receptor
BCRP
OXPHOS
LRRK2
PI4K
CFTR
BTK
Lipase
GTPase
Antifolate
LIM Kinase
PYK2
DNA gyrase
Monoamine Transporter
Xanthine Oxidase
Epoxide Hydrolase
ribosome
Aromatase
MLK
Thyroid hormone receptor(THR)
MicroRNA
ROR
Ligands for Target Protein for PROTAC
Annexin A
PAFR
Vasopressin Receptor
STING
Free radical scavengers
Ephrin Receptor
RSV
GST
SGK
NADPH-oxidase
Arginase
SIK
Glucagon Receptor
Guanylate cyclase
Survivin
Aminopeptidase
PAI-1
FKBP
CRISPR/Cas9
Hydroxylase
Complement System
Neurokinin receptor
Platelet aggregation
IKZF
RAR/RXR
MyD88
Arrestin
Factor Xa
Glucokinase
NAMPT
IRE1
Phosphorylase
MAGL
Cadherin
ATP Citrate Lyase
OAT
ASK
GPX
Protease-activated Receptor
Imidazoline Receptor
NPC1L1
Dynamin
Na+/Ca2+ Exchanger
Bcl-6
AAK1
Glutaminase
NR4A
MTH1
ACK1
Porcupine
AIM2
Decarboxylase
cGAS
Carboxypeptidase
FOXO
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
Transaminase
NEDD8
TOPK
OCT
Cholecystokinin Receptor
Hck
ATG
RANKL/RANK
Amylase
GRK
GlyT
Hexokinase
Bombesin Receptor
PAD
Thrombopoietin Receptor
Orphan Receptor
Wee1
GluCls
CRFR
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Melanocortin Receptor
Aquaporin
GHSR
Adenosine Deaminase
CGRP Receptor
Cuproptosis
Gap Junction Protein
FOXO3
Advanced Glycation End Products
Monocarboxylate transporter
CRM1
gp120/CD4
MIF
VDA
GNRH Receptor
ASCT
Cell Cycle Arrest
LDLR
FLAP
Neuropeptide FF Receptor
Adiponectin Receptor
FABP
Haspin Kinase
AAK1 (AP2 associated kinase 1)
Arp2/3 Complex
Na-K-Cl cotransporter
KSP
Huntingtin
Glutathione reductase
CPT
MELK
Neprilysin
Hippo pathway
p62
Protease
KLF
Oxytocin Receptor
REV-ERB
DAPK
BMI-1
Lysosomal Autophagy
PKM
Taste receptor
CAT
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
Aconitase
Cell wall
CETP
N-Acetylglucosaminyltransferase
CaSR
Photosensitizer
Prolyl Endopeptidase (PREP)
Fas/FasL
Anion Exchanger
Integrase
PROTAC Linker
HCN Channel
Neuropeptide Y Receptor
Somatostatin
Urea Transporter
CD74
hCE
Acetyl-CoA Carboxylase
RXFP receptor
ATTECs
APC/C
Tight Junction Protein
p97

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