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20

Compounds

Cat No. Product Name Synonyms Targets
T77647 Tubulin polymerization-IN-43 Apoptosis , Microtubule Associated
Tubulin polymerization-IN-43 is an inhibitor of tubulin polymerisation.Tubulin polymerization-IN-43 has multiple effects, disrupting the cellular microtubule network by targeting the colchicine locus and promoting cell c...
T77651 Tubulin polymerization-IN-47 Microtubule Associated
Tubulin polymerization-IN-47 is a tubulin polymerization inhibitor and mitotic inhibitor with antitumor activity and inhibitory effects on neuroblastoma cancer cell proliferation, with IC50s of 7 and 12 nM for Chp-134 an...
T77728 Tubulin polymerization-IN-55 Microtubule Associated
Tubulin polymerization-IN-55 is a potent Tubulin Polymerization inhibitor with potential anti-angiogenic and anti-tumour activity, showing anti-proliferative effects against A549, K562, HepG2, MDA-MB-231 and HFL-1.
T61940 Tubulin polymerization-IN-4
Tubulin polymerization-IN-4 is an effective inhibitor of tubulin polymerization (IC50=4.6 μM)。 Tubulin polymerization-IN-4 can destroy tubulin polymerization, block cell cycle at G2/M phase, induce apoptosis, and inhibit...
T72167 Tubulin polymerization-IN-39
Tubulin polymerization-IN-39, a tubulin polymerization inhibitor with an IC50 of 4.9 μM, targets the colchicine-binding site to hinder tubulin polymerization. This compound effectively suppresses cancer cell proliferatio...
T61600 Tubulin polymerization-IN-10
Tubulin polymerization-IN-10 is a highly potent inhibitor of tubulin polymerization, exhibiting an IC50 value of 4.25±0.75 μM. It possesses significant anti-tumor properties [1].
T62040 Tubulin polymerization-IN-30
Tubulin polymerization-IN-30 (compound 6e) is a potent inhibitor of Tubulin polymerization. Tubulin polymerization-IN-30 can disrupt intracellular microtubule organization, arrest cell cycle at the G2/M phase. Tubulin po...
T62217 Tubulin polymerization-IN-9
Tubulin polymerization-IN-9 is a potent inhibitor of tubulin (IC50: 1.82 μM). Tubulin polymerization-IN-9 arrests the cell cycle of K562 cells in G2/M phase and induces apoptosis and mitochondrial depolarization. Tubulin...
T63611 Tubulin polymerization-IN-32
Tubulin polymerization-IN-32 is a tubulin polymerization inhibitor that inhibits the proliferation of cancer cells and can be used to study cancers such as lymphoma.
T80924 Tubulin polymerization-IN-51
Tubulin Polymerization-IN-51 (compound 7u) serves as a tubulin polymerization inhibitor, exhibiting an IC50 range of 2.55 - 17.89μM against SK-Mel-28 cells, and is applicable in cancer research [1].
T60600 Tubulin polymerization-IN-14
Tubulin polymerization-IN-14 (Compound 20a) is a tubulin polymerization inhibitor (IC 50 = 3.15 μM) that exhibits potent anti-vascular and anticancer activities including cancer cell apoptosis [1].
T62349 Tubulin polymerization-IN-8
Tubulin polymerization-IN-8 (compound IIc) is a potent inhibitor of tubulin polymerization that has been demonstrated to concentration-dependently induce cell cycle arrest at the G2/M phase in HCT116 tumor cells. It also...
T80923 Tubulin polymerization-IN-53
Tubulin polymerization-IN-53 (compound 4b) serves as an inhibitor of β-tubulin polymerization and is capable of arresting the cell cycle at the G2/M stage. It demonstrates antiproliferative efficacy against the MDA-MB-23...
T62369 Tubulin polymerization-IN-17
Tubulin aggregation-IN-17 (compound 23g) is a potent inhibitor of tubulin aggregation. tubulin aggregation-IN-17 has a microtubulin-depolymerising effect, induces apoptosis and inhibits migration. tubulin aggregation-IN-...
T62971 Tubulin polymerization-IN-16
Tubulin aggregation-IN-16 (compound 5g) is a potent inhibitor of tubulin aggregation. 16 effectively disrupts microtubule/tubulin dynamics and induces cell cycle arrest at G2/M phase in SGC-7901 cells.
T62477 Tubulin polymerization-IN-18
Tubulin aggregation-IN-18 (compound 3) is a potent tubulin aggregation inhibitor with potential for breast cancer and drug-resistant colon cancer studies.
T61069 Tubulin polymerization-IN-15
Tubulin polymerization-IN-15 (compound 4) is a highly effective inhibitor of tubulin polymerization, with significant potential in cancer research [1].
T60902 Tubulin polymerization-IN-31
Tubulin polymerization-IN-31 (Compound 4c) has antitumor activity and induces apoptosis of cancer cell. Tubulin polymerization-IN-31 is an inhibitor of tubulin polymerization with an IC 50 value of 3.64 μM [1].
T79268 Tubulin polymerization-IN-42
Tubulin polymerization-IN-42 (compound 10j), an indole-substituted furanone, inhibits tubulin polymerization and exhibits anti-cancer properties [1].
T61129 Tubulin polymerization-IN-27
Tubulin polymerization-IN-27 (compound 5j) is an inhibitor of tubulin polymerization. It has the ability to halt the cell cycle specifically at the G2/M phase and also induce apoptosis [1].
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TargetMol