5
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T79207 | SUCNR1-IN-1 | ||
SUCNR1-IN-1 (Compound 20) serves as a potent SUCNR1 inhibitor, exhibiting an IC50 of 88 nM against hSUCNR1. It is utilized in the study of rheumatoid arthritis, liver fibrosis, and obesity [1]. | |||
T81075 | SUCNR1-IN-2 | ||
SUCNR1-IN-2 (Statement 35) serves as an inhibitor of both succinate and succinate receptor 1, utilized in research pertaining to neurodegenerative disorders, including neuroinflammation [1]. | |||
T12216 | NF-56-EJ40 | GPR | |
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM. | |||
T12216L | NF-56-EJ40 hydrochloride | GHSR | |
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride... | |||
T71921 | Cis-Epoxysuccinic acid | ||
Cis-Epoxysuccinic acid, a succinate receptor (SUCNR1/GPR91) agonist, regulates cardiovascular system research by inhibiting cAMP levels with an EC50 value of 2.7 µM. |