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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12939 | SMYD2-IN-1 | Histone Methyltransferase | |
SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM). | |||
T6879 | LLY-507 | LLY507,LLY 507 | Histone Methyltransferase |
LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyltransferase SMYD2. | |||
TQ0100 | AZ505 | Histone Methyltransferase | |
AZ505 is an effective and specific SMYD2 inhibitor (IC50: 0.12 μM). | |||
T7403 | BAY-598 | Histone Methyltransferase | |
BAY-598 is a selective inhibitor of SMYD2 with IC50 values of 27 nM. | |||
T70087 | EPZ032597 | Histone Methyltransferase | |
EPZ032597 is a novel selective inhibitor of SMYD2 with an IC50 of 16 nM. EPZ032597 has anticancer activity and can be used to prevent and treat pancreatic cancer. | |||
T10427 | AZ505 ditrifluoroacetate | Histone Methyltransferase | |
AZ505 ditrifluoroacetate is an effective and selective SMYD2 inhibitor (IC50: 0.12 μM). | |||
T5381 | A-893 | ||
A-893 is a cell-active inhibitor of Methyltransferase SMYD2 (IC 50 = 2.8 nM) . | |||
T63783 | AZ506 | ||
AZ506 is a potent inhibitor of SMYD2 (IC50: 17 nM). AZ506 inhibits SMYD2 methyltransferase activity in cells and reduces SMYD2-mediated methylation signaling. | |||
T26744 | BAY-598 R-isomer | BAY598 R-isomer,BAY 598 R-isomer | |
BAY-598 R-isomer is the R-isomer of BAY589, which is used as a reference compound. It is is an inhibitor of lysine N-methyltransferase (SMYD2) and is selective for SMYD2 over protease-activated receptor 1 (PAR1). |