5
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3987 | Lotamilast | E6005,RVT-501 | PDE |
Lotamilast (RVT-501) is a phosphodiesterase 4 (PDE-4) inhibitor (IC50: 2.8 nM) potentially for the treatment of atopic dermatitis. | |||
T3630 | Relugolix | RVT-601,TAK-385 | GNRH Receptor |
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively bi... | |||
T1774 | Intepirdine | RVT-101,SB 742457,GSK-742457 | 5-HT Receptor |
Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease. | |||
T27154 | Dexelvucitabine | D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC | Reverse Transcriptase |
Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T16779 | Rodatristat ethyl | RVT-014,KAR5585,RVT-1201 | 5-HT Receptor , Hydroxylase |
Rodatristat ethyl (KAR5585) is a first-of-its-kind orally active and potent tryptophan hydroxylase 1 (TPH1) inhibitor that significantly reduces 5-hydroxytryptamine (5-HT) levels and decreases pulmonary arterial hyperten... |