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Search Results for " pdhk1 "

Targets

4

Compounds

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T2028 NG 52 NG52,NG-52,Compound 52 CDK
NG 52 (NG-52) is a cell-permeable, reversible, and ATP-compatible inhibitor of the cell cycle-regulating kinase Cdc28p and the related Pho85p kinase.
T2447 AZD7545 Dehydrogenase
AZD7545 is a potent PDHK inhibitor.
T71147 PBS-1086
PBS-1086 is a novel dual inhibitor of the canonical and noncanonical NF-κB pathways, increasing the magnitude and duration of initial EGFR inhibitor response in multiple NSCLC models, decreasing PDHK1 expression, and sup...
T63012 TM-1
TM-1 is a potent pyruvate dehydrogenase kinase (PDHK) inhibitor that inhibits the activity of PDHK1 (IC50: 2.97 μM) and PDHK2 (IC50: 5.2 μM). TM-1 blocks pyruvate dehydrogenase complex (PDHC) phosphorylation and inhibits...

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-04568 PDK1 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
Pyruvate dehydrogenase kinase, isozyme 1, also known as [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 1, mitochondrial and PDK1, is a member of the PDK / BCKDK protein kinase family. PDK-1 is expressed predominantl...
TargetMol