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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7495 | Hexa-D-arginine | Others | |
Hexa-D-arginine is an inhibitor of furin,blocks the activation of Pseudomonas aeruginosa exotoxin A in vivo. | |||
T83974 | OPC18750 HCl | PDE | |
OPC18750 HCl is a potential phosphodiesterase inhibitor with positive inotropic effects that can be used to study asthma, cancer, diabetes, and psychiatric disorders. | |||
T29112 | VPC171 | VPC 171,VPC-171 | Adenosine Receptor |
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM). | |||
T61274 | PC190723 | ||
PC190723 (Compound 2), an inhibitor of the FtsZ bacterial cell division protein, demonstrates potent efficacy with an IC50 value of 55 ng/ml. Additionally, it showcases notable anti-staphylococcal activity, characterized... | |||
T29109 | VPC12249 | VPC-12249,VPC 12249 | |
VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity. | |||
T24599 | PC170942 Sodium | PC170942 Sodium salt | |
PC170942 Sodium is a water-soluble bacterial cytokinesis inhibitor that acts by inhibiting FtsZ. | |||
TP1160 | Hexa-D-arginine TFA | Furin Inhibitor II TFA | |
Hexa-D-arginine TFA (Furin Inhibitor II TFA) is an inhibitor of furin (Ki values are 0.106, 0.58 and 13.2 μM for furin, PACE4 and PC1 respectively). | |||
TP2038 | Decanoyl-RVKR-CMK | ||
Subtilisin/Kex2p-like proprotein convertase inhibitor; blocks activity of all seven convertases (PC1, PC2, PC4, PACE4, PC5, PC7 and furin). Abolishes proET-1 processing in endothelial cells; inhibits regulated secretion ... | |||
T78224 | Histatin-3 | ||
Histatin-3, a 32-amino-acid peptide, exhibits potent antimicrobial activities and serves as a substrate for proprotein convertase 1 (PC1), where it is primarily cleaved at a site carboxy-terminal to Arg25 (HRGYR↓SN). Add... |