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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5394 | Prulifloxacin | AF 3012,Pruvel,NM441 | Topoisomerase , Antibacterial , Antibiotic |
Prulifloxacin (NM441) is a broad-spectrum fluoroquinolone antibiotic. It Inhibits bacterial DNA synthesis by inhibiting the activity of bacterial DNA topoisomerase II and IV. | |||
T21325 | TAK-441 | TAK441 | Hedgehog/Smoothened |
TAK-441 is an orally active inhibitor of Hedgehog signaling(IC50 = 4.4 nM) with potent antitumor activity. TAK-441 suppresses transcription factor Gli1 mRNA expression and tumor growth. | |||
TP1013 | N-CBZ-Phe-Arg-AMC | Z-FR-AMC | |
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) is a substrate for serine proteases, including cathepsins, kallikrein and plasmin. Absorption/emission of substrate = 330/390 nm (weak fluorescence); absorption/emission of end product (AMC) ... | |||
TP1562 | F1324 | ||
F1324 is a potent, high affinity peptidic inhibitor of B cell lymphoma 6 (BCL6) with an IC50 of 1 nM. F1324 exhibits binding t1/2 value of 441 s and has strong inhibition activity against BCL6 PPI. | |||
T37338 | N-3-oxo-pentanoyl-L-Homoserine lactone | ||
N-3-oxo-pentanoyl-L-Homoserine lactone is a chain-shortened derivative of the bacterial quorum sensing signaling molecule N-3-oxo-octanoyl-L-homoserine lactone .1It inhibits binding of the autoinducer N-3-oxo-hexanoyl ho... |