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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6002 | Enzalutamide | MDV3100 | Androgen Receptor , Autophagy |
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP). Enzalutamide activates autophagy, has antitumor activity, and is commonly used in the treatment of desmoplasia-resistant prostate canc... | |||
T11208 | Enzalutamide-d3 | MDV3100 D3 | Others |
Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells. | |||
T19311 | Enzalutamide carboxylic acid D6 | MDV3100 carboxylic acid D6 | Others |
Enzalutamide carboxylic acid is an inactive metabolite of Enzalutamide. Enzalutamide carboxylic acid D6 is the deuterium labeled Enzalutamide carboxylic acid (MDV3100 carboxylic acid). | |||
T8217 | Enzalutamide carboxylic acid | Androgen Receptor , Drug Metabolite | |
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) . | |||
T19450 | N-desmethyl Enzalutamide | N-desmethyl MDV 3100 | Androgen Receptor |
N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide. N-desmethyl Enzalutamide demonstrates primary and secondary pharmacodynamics of similar p... |