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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T14841 | BVT948 | Phosphatase , P450 , Histone Methyltransferase | |
BVT948 is a protein tyrosine phosphatase (PTP) inhibitor. It can also inhibit several CYP450 isoforms and lysine methyltransferase SETD8 (KMT5A). | |||
T63705 | UNC0379 TFA | ||
UNC0379 TFA is a selective, substrate competitive inhibitor of lysine methyltransferase SETD8 (KMT5A) (IC50: 7.3 μM) and exhibits good selectivity for 15 other methyltransferases. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01584 | PR-Set7 Protein, Human, Recombinant | Human | E. coli |
KMT5A (known as PR-Set7/9, SETD8 and SET8), a member of the SET domain containing methyltransferase family specifically targeting H4K20 for methylation, has been implicated in multiple biological processes. Inhibition of... |