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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13536 | Afoxolaner | Chloride channel , GABA Receptor , Parasite | |
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA & glutamate-regulated uptake of chloride ions, resulting i... | |||
T12770 | RR-11a analog | aza-peptide Michael acceptor, 7a | Parasite |
RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, r... |