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RR-11a analog

RR-11a analog
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Purity:98.64%
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RR-11a analog

Catalog No. T12770Cas No. 685543-66-2
RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.
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Pack SizePriceAvailabilityQuantity
1 mg$213In Stock
5 mg$455In Stock
10 mg$628In Stock
25 mg$1,160In Stock
50 mg$1,980In Stock
100 mg$2,890In Stock
1 mL x 10 mM (in DMSO)$493In Stock
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Product Introduction

Bioactivity
Description
RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.
In vivo
RR-11a analog shows a t1/2 of 3-10 min[2].
Aliasaza-peptide Michael acceptor, 7a
Chemical Properties
Molecular Weight491.49
FormulaC22H29N5O8
Cas No.685543-66-2
Storage & Solubility Information
Storage Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Solubility Information
DMSO: 112.5 mg/mL (228.9 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0346 mL10.1731 mL20.3463 mL101.7315 mL
5 mM0.4069 mL2.0346 mL4.0693 mL20.3463 mL
10 mM0.2035 mL1.0173 mL2.0346 mL10.1731 mL
20 mM0.1017 mL0.5087 mL1.0173 mL5.0866 mL
50 mM0.0407 mL0.2035 mL0.4069 mL2.0346 mL
100 mM0.0203 mL0.1017 mL0.2035 mL1.0173 mL

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