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RR-11a analog

RR-11a analog
RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.
Catalog No. T12770Cas No. 685543-66-2
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Purity:98.64%
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RR-11a analog

Catalog No. T12770Cas No. 685543-66-2

RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.
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Pack SizePriceAvailabilityQuantity
1 mg$213In Stock
5 mg$455In Stock
10 mg$628In Stock
25 mg$1,160In Stock
50 mg$1,980In Stock
100 mg$2,890In Stock
1 mL x 10 mM (in DMSO)$493In Stock
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Product Introduction

Bioactivity
Description
RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.
Targets&IC50
AE (ixodes ricinus):4.5 nM , AE1 (Trichomonas Vaginalis):4.5 nM , AE (Schistosoma mansoni):31 nM
In vivo
RR-11a analog shows a t1/2 of 3-10 min[2].
Aliasaza-peptide Michael acceptor, 7a
Chemical Properties
Molecular Weight491.49
FormulaC22H29N5O8
Cas No.685543-66-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 112.5 mg/mL (228.9 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0346 mL10.1731 mL20.3463 mL101.7315 mL
5 mM0.4069 mL2.0346 mL4.0693 mL20.3463 mL
10 mM0.2035 mL1.0173 mL2.0346 mL10.1731 mL
20 mM0.1017 mL0.5087 mL1.0173 mL5.0866 mL
50 mM0.0407 mL0.2035 mL0.4069 mL2.0346 mL
100 mM0.0203 mL0.1017 mL0.2035 mL1.0173 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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