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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $213 | In Stock | |
5 mg | $455 | In Stock | |
10 mg | $628 | In Stock | |
25 mg | $1,160 | In Stock | |
50 mg | $1,980 | In Stock | |
100 mg | $2,890 | In Stock | |
1 mL x 10 mM (in DMSO) | $493 | In Stock |
Description | RR-11a analog (aza-peptide Michael acceptor, 7a) is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively. |
Targets&IC50 | AE (ixodes ricinus):4.5 nM , AE1 (Trichomonas Vaginalis):4.5 nM , AE (Schistosoma mansoni):31 nM |
In vivo | RR-11a analog shows a t1/2 of 3-10 min[2]. |
Alias | aza-peptide Michael acceptor, 7a |
Molecular Weight | 491.49 |
Formula | C22H29N5O8 |
Cas No. | 685543-66-2 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 112.5 mg/mL (228.9 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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