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Search Results for " he1 "

Targets

9

Compounds

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
TP2239L [D-Phe12]-Bombesin acetate [D-Phe12]-Bombesin acetate(108437-87-2 free base) Bombesin Receptor
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
TP1916L1 [D-Phe12,Leu14]-Bombesin acetate [D-Phe12,Leu14]-Bombesin acetate(108437-88-3 Free base) Bombesin Receptor
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
TP1987 [Nphe1]Nociceptin(1-13)NH2
Selective and competitive nociceptin receptor antagonist, devoid of any agonist activity. Binds selectively to recombinant nociceptin receptors (pKi = 8.4), and competitively antagonizes the actions of nociceptin in vitr...
TP1988 [Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2
Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo. Selective, competitive antagonism at the nociceptin receptor has also been reported (pA2 = 7.02 and 6.75 in the guinea pig ileum a...
TP1916 [D-Phe12,Leu14]-Bombesin
Bombesin receptor antagonist that inhibits bombesin binding to rat brain with an IC50 value of 2 μM. Inhibits amylase release in vitro (IC50 = 4 μM) and attenuates bombesin-mediated suppression of food intake in vivo.
T76632 (Phe13,Tyr19)-MCH (human, mouse, rat)
(Phe13,Tyr19)-MCH (human, mouse, rat) serves as a potent ligand for SLC-1 and S643b receptors and can act as an agonist for these receptors [1].
T75909 [Nphe1]Nociceptin(1-13)NH2 TFA
[Nphe1]Nociceptin(1-13)NH2 is a novel endogenous ligand for the nociceptin/orphanin FQ (NC) receptor, acting as a selective and competitive antagonist without any agonist effects. It binds specifically to recombinant noc...
TP2239 [D-Phe12]-Bombesin Others
Bombesin receptor antagonist
T76602 (D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1a on Luteinizing hormone (LH) production [1].

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-01114 NPC2 Protein, Human, Recombinant (His) Human HEK293
Niemann-Pick Type C2 (NPC2) plays an important role in the regulation of intracellular cholesterol homeostasis via direct binding with free cholesterol. NPC2 is an intralysosomal protein that binds cholesterol in vitro. ...
TMPY-04990 NPC2 Protein, Mouse, Recombinant (His) Mouse HEK293
Niemann-Pick Type C2 (NPC2) plays an important role in the regulation of intracellular cholesterol homeostasis via direct binding with free cholesterol. NPC2 is an intralysosomal protein that binds cholesterol in vitro. ...
TMPY-03658 ETHE1 Protein, Human, Recombinant (His) Human E. coli
ETHE1, also known as HSCO, is a sulfur dioxygenase that localizes within the mitochondrial matrix. ETHE1 probably plays an important role in metabolic homeostasis in mitochondria. It may also function as a nuclear-cytopl...
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