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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0702 | Gabapentin | Neurontin,Gabapentine,Aclonium | Calcium Channel , GABA Receptor |
Gabapentin (Neurontin) is an Anti-epileptic Agent. The physiologic effect of gabapentin is by means of Decreased Central Nervous System Disorganized Electrical Activity. | |||
T6507 | Gabapentin hydrochloride | Neurontin HCl,Gabapentin HCl | Calcium Channel , GABA Receptor |
Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain. | |||
T15366 | Gabapentin enacarbil | XP-13512 | Others , Calcium Channel |
Gabapentin enacarbil (XP-13512) is a prodrug for the anticonvulsant and analgesic drug gabapentin. Gabapentin enacarbil provides sustained dose-proportional exposure to gabapentin and predictable bioavailability. | |||
T28346 | PD-217014 HCl | PD 217014,PD217014,PD-217,014,PD-217014 | |
PD-217014 is a GABA analog. It inhibits (3)H-gabapentin binding to alpha(2)delta subunit of voltage-gated calcium channels in a concentration-dependent manner (K(i) = 18 nmol/l). PD-217014 possesses visceral analgesic ac... | |||
T30188 | Atagabalin | PD 0200390,PD-0200390,PD0200390 | |
Atagabalin, also known as PD 0200390, is a gabamimetic agent under development for the treatment for insomnia. Atagabalin is related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was disc... | |||
T71206 | Tiagabine-d6 hydrochloride | ||
Tiagabine-d6 is intended for use as an internal standard for the quantification of tiagabine by GC- or LC-MS. Tiagabine is an inhibitor of GABA transporter 1. It inhibits seizures induced by DMCM in mice. Tiagabine reduc... |