3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1906 | Molibresib | GSK 525762A,GSK525762,I-BET 762 | Epigenetic Reader Domain |
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM). | |||
T11472L | Molibresib besylate | I-BET 762 besylate,GSK 525762C | CCR |
Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM). | |||
T11472 | GSK 525768A | Others | |
GSK 525768A, the inactive enantiomer of GSK525762A, exhibits no activity towards BET. |