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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4664 | ML 297 | ML297 | Potassium Channel |
ML 297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator (IC50 values are 160, 887 and 914 nM for GIRK1/2, GIRK1/4 and GIRK1/3 respectively). ML 297 exhibits no effect on GIRK2, GIRK2/3, Kir2.1 and Kv7.4 channels, an... | |||
T7899 | VU0810464 | Potassium Channel | |
VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK, Kir3) activator. | |||
T17246 | VU0529331 | Others | |
VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel activator (EC50s: 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively). It is also effectiv... | |||
T27502 | Gue1654 | Gue-1654,Gue 1654 | |
Gue1654 is a modulator of oxoeicosanoid receptor 1 (OXE-R). Gue1654 selectively inhibits Gβγ upon activation of the Gαi-βγ heterotrimer by OXE-R. Gue1654 inhibits Gβγ-mediated opening of GIRK1/2 channels in HEK293 cells. |