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Search Results for " ffa2 "

11

Compounds

Cat No. Product Name Synonyms Targets
T3171 GSK137647A GSK 137647 GPR
GSK137647A (GSK 137647) is a selective FFA4 agonist.
T71177 LCRF-0004
LCRF-0004 is a potent and selective RON receptor tyrosine kinase inhibitor. The RON receptor tyrosine kinase has been identified as an important mediator of KRAS oncogene addiction and is overexpressed in the majority o...
T15388 GLPG0974 GLPG-0974 GPR
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
T8642 4-CMTB GPR
4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).
T60184 TUG-499 GPR , PPAR
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 has an affinity for FFAR1 or GPR40 over the related receptors FFA2, FFA3 and the nuclear receptor PPARγ, as well as other di...
T7796 TUG-1375 GPR
TUG-1375 is an Agonist of Thiazolidine Free Fatty Acid Receptor 2
T71179 LON63114
LON63114, also known as FFA2-Agonist-1 is a selective orthosteric agonist of human FFA2. FFA2-Agonist-1 is potentially useful in the treatment of gastrointestinal disorders and inflammatory bowel diseases. LON63114 was ...
T34966 TUG-1609
TUG-1609 is a fluorescent tracer of FFA2 with good spectral properties and high affinity.
T23877 CFMB
CFMB is the FFA2 receptor agonist.
T37896 AZ 1729
FFA2 allosteric agonist. Inhibits forskolin-induced cAMP increase and stimulates 35SGTPγS binding in biochemical assays (pEC50 values are 6.9 and 7.23, respectively). Binds at allosteric binding site. In functional assay...
T83955 MOMBA
MOMBA is a selective orthosteric agonist specifically targeting engineered human free fatty acid 2 (hFFA2) receptors, particularly those modified as designer receptors activated by designer drugs (DREADD). It demonstrate...
TargetMol