5
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T71848 | DS1 | ||
DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse. | |||
T11103 | DS18561882 | Others | |
DS18561882 also inhibited MTHFD1 (IC50=0.57).DS18561882 had good oral drug kinetics.DS18561882 is a potent isozyme-selective methylene tetrahydrofolate dehydrogenase 2 (MTHFD2) inhibitor with IC50 value of 0.0063. | |||
T60681 | DS12881479 | MNK | |
DS12881479 can be used in cancer research which is a potent and selective inhibitor of Mnk1(IC 50 =21 nM) [1]. | |||
T11102 | DS16570511 | Calcium Channel | |
DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter. It effectively blocks the increase in Ca2+ influx dependent on MCU or MICU1 [1]. | |||
T63196 | DS17701585 | ||
DS17701585 is an orally active, selective inhibitor of EP300 and CBP, capable of acting on CBP (IC50: 0.040 μM), EP300 (IC50: 0.15 μM), H3K27 (IC50: 0.45 μM) and SOX2 (IC50: 0.7 μM), and can be used to study cancer. |