carm1-in-1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T10682L	CARM1-IN-1	CARM1-IN-7G	Histone Methyltransferase
	CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM.		Histone Methyltransferase
T64186	CARM1-IN-1 hydrochloride
	CARM1-IN-1 hydrochloride is a potent and selective inhibitor of CARM1 (IC50: 8.6 μM) with low inhibition of PRMT1 and SET7.
T4013	SGC2085 HCl		Histone Methyltransferase
	SGC2085 is a potent and selective coactivator associated arginine methyltransferase 1 (CARM1) Inhibitor with an IC50 of 50 nM and more than undred-fold selectivity over other PRMTs. CARM1 is an important positive modulat...		Histone Methyltransferase
T79007	CARM1-IN-3		Histone Methyltransferase
	CARM1-IN-3 (compound 17b) is a potent, selective inhibitor of co-activator associated arginine methyltransferase (CARM1), exhibiting IC50 values of 0.07 µM for CARM1 and greater than 25 µM for CARM3 [1].		Histone Methyltransferase