Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 < 600 μM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 38.00 | |
2 mg | In stock | $ 54.00 | |
5 mg | In stock | $ 89.00 | |
10 mg | In stock | $ 162.00 | |
25 mg | In stock | $ 297.00 | |
50 mg | In stock | $ 547.00 | |
100 mg | In stock | $ 779.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 109.00 |
Description | CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM. |
In vitro | In human LNCaP cells, CARM1-IN-1 significantly reduces the PSA promoter activity in a dose-dependent manner[1]. |
Synonyms | CARM1-IN-7G |
Molecular Weight | 555.26 |
Formula | C26H21Br2NO3 |
CAS No. | 1020399-49-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 30 mg/mL (54 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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CARM1-IN-1 1020399-49-8 Chromatin/Epigenetic Histone Methyltransferase CARM1-IN-7G inhibitor inhibit