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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T35348 | LDN-193189 2HCl | LDN-193189 2HCl,DM-3189 2HCl | ALK , TGF-beta/Smad |
LDN-193189 2HCl (DM-3189 2HCl) is a selective BMP signaling inhibitor that inhibits ALK1,ALK2,ALK3 and ALK6, showing IC50s of 0.8 nM, 0.8 nM, 5.3 nM, and 16.7 nM, respectively, in kinase assays.LDN-193189 2HCl inhibited ... | |||
T6158 | LDN-193189 HCl | LDN193189 Hydrochloride | ALK |
LDN-193189 HCl (LDN193189 Hydrochloride) is a selective BMP type I receptor kinases inhibitor. | |||
T63897 | LDN193189 Tetrahydrochloride | ||
LDN193189 Tetrahydrochloride is a selective inhibitor of BMPI-type receptors and inhibits ALK2 (IC50: 5 nM) and ALK3 (IC50: 30 nM), with weak effects on ALK4, ALK5 and ALK7 (IC50 ≥ 500 nM). | |||
T1935 | LDN193189 | LDN-193189,DM-3189,LDN 193189 | ALK , TGF-beta/Smad |
LDN193189 (LDN-193189) (DM 3189) is a selective BMP signaling inhibitor, inhibiting the transcriptional activity of ALK2 and ALK3 (IC50s: 0.8/0.8/5.3/16.7 nM for ALK1/2/3/6). |