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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T13456 | (S)-Willardiine | (-)-Willardiine,L-willardiine,Willardiine | iGluR |
(S)-Willardiine (L-willardiine) is present in the seeds of Acacia and Mimosa. (S)-Willardiine is an AMPA/kainate receptor agonist (EC50 = 44.8 μM). | |||
T50094 | DL-Willardiine | 2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid | Others |
DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate. It is an agonist of mGluR5, which regulates the activity of enzymes involved in... | |||
T13394 | ZEN-3862 | ZEN3862,ZEN 3862 | Epigenetic Reader Domain |
ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4. |