Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 97.00 | |
2 mg | In stock | $ 139.00 | |
5 mg | In stock | $ 228.00 | |
10 mg | In stock | $ 355.00 | |
25 mg | In stock | $ 628.00 | |
50 mg | In stock | $ 888.00 | |
100 mg | In stock | $ 1,190.00 | |
500 mg | In stock | $ 2,390.00 |
Description | ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4. |
Targets&IC50 | BRD4 BD2:, BRD4 BD1:0.16 μM |
Synonyms | ZEN3862, ZEN 3862 |
Molecular Weight | 340.35 |
Formula | C19H17FN2O3 |
CAS No. | 1952264-33-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Soluble
You can also refer to dose conversion for different animals. More
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ZEN-3862 1952264-33-3 Chromatin/Epigenetic Epigenetic Reader Domain ZEN3862 ZEN 3862 inhibitor inhibit