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Regrelor disodium

Name: Regrelor disodium
Brand: TargetMol
SKU: T34280
Price: 82 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T34280Cas No. 676251-22-2

Alias Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589

Regrelor disodium (INS 50589) is a P2Y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, curbs cell proliferation, and reduces inflammation.

Regrelor disodium

🥰Excellent

Purity: 99.95%

Catalog No. T34280Alias Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589Cas No. 676251-22-2

Pack Size	Price	Availability
1 mg	$82	In Stock
5 mg	$181	In Stock
10 mg	$267	In Stock
25 mg	$413	In Stock
50 mg	$571	In Stock
100 mg	$763	In Stock
200 mg	$1,030	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.95%

ee:100%

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COA CSFC HNMR LCMS ORP

Product Introduction

Bioactivity

Description	Regrelor disodium (INS 50589) is a P2Y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, curbs cell proliferation, and reduces inflammation.
Synonyms	Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589

Chemical Properties

Molecular Weight	576.41
Formula	C₂₂H₂₃N₆Na₂O₈P
Cas No.	676251-22-2
Smiles	[O-]P(OC[C@H]1O[C@H]([C@]2([C@@]1(O[C@H](/C=C/C3=CC=CC=C3)O2)[H])[H])N4C5=NC=NC(NC(NCC)=O)=C5N=C4)([O-])=O.[Na+].[Na+]
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 105 mg/mL (182.16 mM), Sonication is recommended.

DMSO: < 1 mg/mL (insoluble or slightly soluble)

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	1.7349 mL	8.6744 mL	17.3488 mL	86.7438 mL
5 mM	0.3470 mL	1.7349 mL	3.4698 mL	17.3488 mL
10 mM	0.1735 mL	0.8674 mL	1.7349 mL	8.6744 mL
20 mM	0.0867 mL	0.4337 mL	0.8674 mL	4.3372 mL
50 mM	0.0347 mL	0.1735 mL	0.3470 mL	1.7349 mL
100 mM	0.0173 mL	0.0867 mL	0.1735 mL	0.8674 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc