Powder: -20°C for 3 years | In solvent: -80°C for 1 year
UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 47.00 | |
10 mg | In stock | $ 80.00 | |
25 mg | In stock | $ 146.00 | |
50 mg | In stock | $ 247.00 | |
100 mg | In stock | $ 372.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 52.00 |
Description | UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. |
Targets&IC50 | SETD8:7.3 μM |
In vitro | UNC0379 is competitive with the peptide substrate and noncompetitive with the cofactor SAM. [1] |
Molecular Weight | 413.56 |
Formula | C23H35N5O2 |
CAS No. | 1620401-82-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 76 mg/mL (183.8 mM)
H2O: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
UNC0379 1620401-82-2 Chromatin/Epigenetic Histone Methyltransferase UNC-0379 neuroblastoma lysine methyltransferase pulmonary fibrosis antitumor UNC 0379 Inhibitor OVCAR3 HGSOC Ovarian cancer inhibit JHOS3 inhibitor