keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Thalidomide-O-amido-PEG2-C2-NH2 TFA (E3 Ligase Ligand-Linker Conjugates 24 TFA) is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-O-amido-PEG2-C2-NH2 TFA incorporates the Thalidomide based cereblon ligand and 2-unit PEG linker used in PROTAC technology.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 33.00 | |
2 mg | In stock | $ 47.00 | |
5 mg | In stock | $ 75.00 | |
10 mg | In stock | $ 108.00 | |
25 mg | In stock | $ 183.00 | |
50 mg | In stock | $ 272.00 | |
100 mg | In stock | $ 396.00 | |
200 mg | In stock | $ 743.00 | |
500 mg | In stock | $ 1,450.00 |
Description | Thalidomide-O-amido-PEG2-C2-NH2 TFA (E3 Ligase Ligand-Linker Conjugates 24 TFA) is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-O-amido-PEG2-C2-NH2 TFA incorporates the Thalidomide based cereblon ligand and 2-unit PEG linker used in PROTAC technology. |
In vitro | PROTACs contain two different ligands connected by a linker; one of them is a ligand for an E3 ubiquitin ligase and the other one is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins[1]. |
Synonyms | E3 Ligase Ligand-Linker Conjugates 24 TFA, Cereblon Ligand-Linker Conjugates 10 TFA |
Molecular Weight | 576.48 |
Formula | C23H27F3N4O10 |
CAS No. | 1957235-75-4 |
keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 150 mg/mL (260.20 mM)
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Thalidomide-O-amido-PEG2-C2-NH2 TFA 1957235-75-4 Others PROTAC E3 Ligase Ligand-Linker Conjugate Thalidomide O amido PEG2 C2 NH2 TFA Cereblon Ligand-Linker Conjugates 10 E3 Ligase Ligand-Linker Conjugates 24 E3 Ligase Ligand-Linker Conjugates 24 TFA Inhibitor Cereblon Ligand-Linker Conjugates 10 TFA inhibit Thalidomide-O-amido-PEG-2-C2-NH2 TFA ThalidomideOamidoPEG2C2NH2 TFA E3 Ligase Ligand-Linker Conjugates inhibitor