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TG6-10-1

Catalog No. T2428   CAS 1415716-58-3

TG6-10-1 is an EP2 antagonist.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
TG6-10-1 Chemical Structure
TG6-10-1, CAS 1415716-58-3
Pack Size Availability Price/USD Quantity
1 mg In stock $ 48.00
2 mg In stock $ 69.00
5 mg In stock $ 117.00
10 mg In stock $ 157.00
25 mg In stock $ 498.00
50 mg In stock $ 928.00
100 mg In stock $ 1,200.00
1 mL * 10 mM (in DMSO) In stock $ 131.00
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Purity: 100%
Purity: 99.11%
Purity: 98%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description TG6-10-1 is an EP2 antagonist.
Kinase Assay Rac Activity Assays: Rac activity is determined from lysates of the MDA-MB-435 and MDA-MB-231 human metastatic cancer cell lines (from ATCC). Cancer cells in culture medium (DMEM, 10% FBS, pH 7.5) are treated with vehicle (0.1% DMSO) or varying concentrations of EHop-016 (0–10 μM) for 24 h. Rac1 activity is determined using the G-LISA Rac1 activation assay kit.
Molecular Weight 448.43
Formula C23H23F3N2O4
CAS No. 1415716-58-3

Storage

store under nitrogen

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 60 mg/mL (133.8 mM)

TargetMolReferences and Literature

1. Jiang J, et al. Proc Natl Acad Sci U S A. 2013 Feb 26;110(9):3591-3596.

Related compound libraries

This product is contained In the following compound libraries:
Anti-Neurodegenerative Disease Compound Library Bioactive Compound Library Fluorochemical Library Anti-Obesity Compound Library Inhibitor Library Anti-Parkinson's Disease Compound Library NO PAINS Compound Library Target-Focused Phenotypic Screening Library Immunology/Inflammation Compound Library Neurotransmitter Receptor Compound Library

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Keywords

TG6-10-1 1415716-58-3 GPCR/G Protein Immunology/Inflammation Neuroscience 5-HT Receptor Prostaglandin Receptor TG-6-10-1 TG6101 Inhibitor Serotonin Receptor inhibit TG6 10 1 5-hydroxytryptamine Receptor inhibitor

 

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