Powder: -20°C for 3 years
In solvent: -80°C for 6 months
Sparsentan is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM, respectively)
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | 126.00 | |
10 mg | In stock | 207.00 | |
25 mg | In stock | 369.00 | |
50 mg | In stock | 612.00 | |
100 mg | In stock | 1017.00 | |
1 mL * 10 mM (in DMSO) | In stock | 207.00 |
Description | Sparsentan is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM, respectively) |
Targets&IC50 | Human angiotensin II , Human endothelin A , Rat angiotensin II , angiotensin II receptor , Endothelin A receptor |
Synonyms | RE-021 , DARA-a |
Purity | 98.81% |
Molecular Weight | 592.8 |
Formula | C32H40N4O5S |
CAS No. | 254740-64-2 |
Powder: -20°C for 3 years
In solvent: -80°C for 6 months
DMSO: 240 mg/mL (404.89 mM), Need ultrasonic
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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