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Regrelor disodium

Name: Regrelor disodium
Brand: TargetMol
SKU: T34280
Price: 82 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T34280Cas No. 676251-22-2

Alias Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589

Regrelor disodium (INS 50589) is a P2Y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, curbs cell proliferation, and reduces inflammation.

Regrelor disodium

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Purity: 99.89%

Catalog No. T34280Alias Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589Cas No. 676251-22-2

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$82	In Stock	In Stock
5 mg	$181	In Stock	In Stock
10 mg	$267	In Stock	In Stock
25 mg	$413	In Stock	In Stock
50 mg	$571	In Stock	In Stock
100 mg	$763	In Stock	In Stock
200 mg	$1,030	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.89%

ee:100%

Appearance:Solid

Color:White

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COA CSFC HNMR ORP LCMS

Product Introduction

Bioactivity

Description	Regrelor disodium (INS 50589) is a P2Y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, curbs cell proliferation, and reduces inflammation.
Synonyms	Regrelor sodium, Regrelor, INS-50589, INS50589, INS 50589

Chemical Properties

Molecular Weight	576.41
Formula	C₂₂H₂₃N₆Na₂O₈P
Cas No.	676251-22-2
Smiles	[O-]P(OC[C@H]1O[C@H]([C@]2([C@@]1(O[C@H](/C=C/C3=CC=CC=C3)O2)[H])[H])N4C5=NC=NC(NC(NCC)=O)=C5N=C4)([O-])=O.[Na+].[Na+]
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 105 mg/mL (182.16 mM), Sonication is recommended.

DMSO: < 1 mg/mL (insoluble or slightly soluble)

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	1.7349 mL	8.6744 mL	17.3488 mL	86.7438 mL
5 mM	0.3470 mL	1.7349 mL	3.4698 mL	17.3488 mL
10 mM	0.1735 mL	0.8674 mL	1.7349 mL	8.6744 mL
20 mM	0.0867 mL	0.4337 mL	0.8674 mL	4.3372 mL
50 mM	0.0347 mL	0.1735 mL	0.3470 mL	1.7349 mL
100 mM	0.0173 mL	0.0867 mL	0.1735 mL	0.8674 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc