Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Pim1/AKK1-IN-1 (LKB1/AAK1 dual inhibitor) is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 82.00 | |
2 mg | In stock | $ 133.00 | |
5 mg | In stock | $ 193.00 | |
10 mg | In stock | $ 292.00 | |
25 mg | In stock | $ 515.00 | |
50 mg | In stock | $ 747.00 | |
100 mg | In stock | $ 1,050.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 213.00 |
Description | Pim1/AKK1-IN-1 (LKB1/AAK1 dual inhibitor) is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. |
Targets&IC50 | LKB1:380 nM (Kd), Pim1:35 nM (Kd), MST2:75 nM (Kd), AKK1:53 nM (Kd) |
Synonyms | LKB1/AAK1 dual inhibitor, MDK-2275 |
Molecular Weight | 339.35 |
Formula | C20H13N5O |
CAS No. | 1093222-27-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 15 mg/mL (44.2 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Pim1/AKK1-IN-1 1093222-27-5 Chromatin/Epigenetic JAK/STAT signaling Stem Cells Pim Hippo pathway Pim kinases Pim1/AKK1IN1 MDK 2275 Pim-1/AKK1-IN-1 inhibit LKB1/AAK1 dual inhibitor MDK-2275 Inhibitor Pim1/AKK1 IN 1 MDK2275 inhibitor