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LY 517717

Catalog No. T27920 CAS 313489-71-3

Synonyms: LY-517717, LY517717

LY 517717 is an orally active inhibitor of coagulation factor Xa with antithrombotic activity for the study of venous thromboembolism (VTE).

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LY 517717, CAS 313489-71-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 293.00
5 mg	In stock	$ 722.00
10 mg	In stock	$ 987.00
25 mg	In stock	$ 1,520.00
50 mg	In stock	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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Purity: 99.88%

ee: 99.64%

Biological Description

Chemical Properties

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Description

LY 517717 is an orally active inhibitor of coagulation factor Xa with antithrombotic activity for the study of venous thromboembolism (VTE).

Synonyms	LY-517717, LY517717
Molecular Weight	459.58
Formula	C27H33N5O2
CAS No.	313489-71-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Agnelli G, et al. A phase II study of the oral factor Xa inhibitor LY517717 for the prevention of venous thromboembolism after hip or knee replacement. J Thromb Haemost. 2007 Apr;5(4):746-53. 2. Eriksson BI,et al. Comparative pharmacodynamics and pharmacokinetics of oral direct thrombin and factor xa inhibitors in development. Clin Pharmacokinet. 2009;48(1):1-22. 3. Eriksson BI, et al. Oral anticoagulants in development: focus on thromboprophylaxis in patients undergoing orthopaedic surgery. Drugs. 2006;66(11):1411-29. 4. Talele TT, et al. Successful applications of computer aided drug discovery: moving drugs from concept to the clinic. Curr Top Med Chem. 2010;10(1):127-41.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

LY 517717 313489-71-3 Metabolism Factor Xa LY-517717 LY517717 inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.