Powder: -20°C for 3 years
In solvent: -80°C for 2 years
Ceefourin 1 is a highly selective multidrug resistance protein 4 (<a href="/target/MRP" style="display: inline; color: #c13a36">MRP</a>4) inhibitor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 59.00 | |
5 mg | In stock | $ 85.00 | |
10 mg | In stock | $ 126.00 | |
25 mg | In stock | $ 263.00 | |
50 mg | In stock | $ 409.00 | |
100 mg | In stock | $ 774.00 | |
200 mg | In stock | $ 1,161.00 |
Description | Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor. |
In vitro | Ceefourin 1 and Ceefourin 2, that inhibit transport of a broad range of MRP4 substrates, yet are highly selective for MRP4 over other ABC transporters, including P-glycoprotein (P-gp), ABCG2 (Breast Cancer Resistance Protein;?BCRP) and MRP1 (multidrug resistance protein 1;?ABCC1).?Both compounds are more potent MRP4 inhibitors in cellular assays than the most widely used inhibitor, MK-571, requiring lower concentrations to effect a comparable level of inhibition.?Furthermore, Ceefourin 1 and Ceefourin 2 have low cellular toxicity, and high microsomal and acid stability. |
Molecular Weight | 294.41 |
Formula | C11H10N4S3 |
CAS No. | 315702-40-0 |
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
DMSO: 10 mM
( < 1 mg/ml refers to the product slightly soluble or insoluble )
You can also refer to dose conversion for different animals. More
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Ceefourin 1 315702-40-0 Immunology/Inflammation MRP P-glycoprotein chemosensitizers inhibit efflux protein resistance Ceefourin1 MRP4 HEK293 D-luciferin ABC ABCG2 P-gp multidrug MRP1 Inhibitor neuroblastoma Ceefourin-1 ABCC1 BCRP inhibitor