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Betahistine dihydrochloride

Catalog No. T0246 CAS 5579-84-0

Synonyms: Betahistine 2HCl, PT-9

Betahistine hydrochloride is a histamine analog and H1 receptor agonist that serves as a vasodilator.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Betahistine dihydrochloride, CAS 5579-84-0

Pack Size	Availability	Price/USD
50 mg	In stock	$ 30.00
100 mg	In stock	$ 42.00
1 g	In stock	$ 50.00
1 mL * 10 mM (in DMSO)	In stock	$ 46.00

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Purity: 99.88%

Purity: 99.34%

Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Betahistine hydrochloride is a histamine analog and H1 receptor agonist that serves as a vasodilator.
Targets&IC50	Histamine H3 receptor:1.9 μM

Synonyms	Betahistine 2HCl, PT-9
Molecular Weight	209.12
Formula	C8H14Cl2N2
CAS No.	5579-84-0

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 2 years

Solubility Information

DMSO: 36 mg/mL (172.1 mM)

H2O: 35 mg/mL (167.4 mM)

Ethanol: 1 mg/mL (4.78 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Gbahou F, et al. J Pharmacol Exp Ther, 2010, 334(3), 945-954. 2. Mira E, et al. Eur Arch Otorhinolaryngol, 2003, 260(2), 73-77. 3. Strupp M, et al. Acta Otolaryngol, 2008, 128(5), 520-524. 4. Tighilet B, et al. Eur J Pharmacol, 2002, 446(1-3), 63-73.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Obesity Compound Library FDA-Approved & Pharmacopeia Drug Library Target-Focused Phenotypic Screening Library Drug Repurposing Compound Library Immunology/Inflammation Compound Library Bioactive Compounds Library Max NMPA-Approved Drug Library GPCR Compound Library Neuronal Signaling Compound Library NO PAINS Compound Library

Related Products

Related compounds with same targets

Noberastine Enerisant HCl Linetastine Impromidine hydrochloride Talastine Donetidine Oxatomide Dalcotidine

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

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