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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9459 | GR103545 | Others | |
GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging. | |||
T77374 | Ontuxizumab | MORAb-004 | Others |
Ontuxizumab (MORAb-004) is a monoclonal antibody targeting endomelanic acid with anti-tumor effects.Ontuxizumab is a potent IgG1/κ anti-endothelin (TEM-1 or CD248) monoclonal antibody for the treatment of metastatic mela... | |||
T69475 | Dinalbuphine sebacate | ||
Dinalbuphine sebacate is a long-lasting prodrug of nalbuphine, acting as a moderate-efficacy partial agonist or antagonist of the μ-opioid receptor and as a high-efficacy partial agonist of the κ-opioid receptor. | |||
T81297 | Renvistobart | ||
Renvistobart is a monoclonal antibody belonging to the immunoglobulin G1-κ class, targeting the human T cell immunoreceptor with Ig and ITIM domains (TIGIT, also known as VSIG9 or VSTM3) [1]. | |||
T40510 | Ac-RYYRWK-NH2 TFA | Ac-RYYRWK-NH2 TFA | |
Ac-RYYRWK-NH2 is a highly effective and specific partial agonist for the nociceptin receptor (NOP). It demonstrates a remarkable affinity for rat cortical membranes ORL1, with [3H]Ac-RYYRWK-NH2 exhibiting a Kd value of 0... | |||
T71491 | Enadoline (Free Base) | ||
Enadoline (Free Base) is a kappa-opioid receptor agonist; PD 129290 (CAM 570; CI 977) is the S,S(-)-enantiomer; PD 129289 (CAM 569) is the corresponding R,R(+)-enantiomer. In human studies, it produced visual distortions... | |||
T83913 | Mitraciliatine | ||
Mitraciliatine, an alkaloid discovered in M. speciosa (Kratom in Thai), acts as a partial agonist for the μ-opioid receptor (MOR) and an agonist for the κ-opioid receptor (KOR), demonstrating selectivity for these recept... | |||
T72696 | UCK2 Inhibitor-3 | ||
UCK2 Inhibitor-3 is a non-competitive inhibitor targeting uridine-cytidine kinase 2 (UCK2), a key enzyme in the pyrimidine salvage pathway, with an IC50 value of 16.6 μM. Notably, UCK2 can partially substitute for dihydr... |